SCHEMBL4050906

SCHEMBL4050906

O=C(NC1(C(=O)N2CCC3C2C(=O)CN3C(=O)Cc2cccnc2)CCCCC1)Oc1cc2sccc2s1

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PAX8 Q06710 1/20 0.32
GPR132 Q9UNW8 1/20 0.32
OPRM1 P35372 1/20 0.31
OPRK1 P41145 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TNKS O95271 1/20 0.30
PARP1 P09874 1/20 0.30
PARP2 Q9UGN5 1/20 0.30
PARP4 Q9UKK3 1/20 0.30
PARP3 Q9Y6F1 1/20 0.30
TACR2 P21452 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
NAMPT P43490 2/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4048915 0.87 SMYD3 (0.34) GPR132
SCHEMBL4042619 0.84 HPGD (0.33) SMN1; SMN2
SCHEMBL4048571 0.83 MEN1 (0.32)
SCHEMBL4046730 0.82 CTSL (0.36) SMN1; SMN2
SCHEMBL4042884 0.81 CTSK (0.41) PAX8ALDH1A1
SCHEMBL4051435 0.81 HTRA1 (0.33) PAX8GPR132TNKSPARP1PARP2
SCHEMBL4038641 0.81 CTSK (0.33) PAX8GPR132ALDH1A1TNKSPARP1
SCHEMBL4043944 0.80 CTSK (0.33) PAX8ALDH1A1
SCHEMBL4041874 0.79 CHRNB2 (0.37) PAX8SMN1; SMN2NAMPT
SCHEMBL4048563 0.78 HDAC1 (0.40) GPR132

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed