SCHEMBL4052843

SCHEMBL4052843

CC(C)(C)[C@H](NC(=O)c1cc2cc(F)ccc2[nH]1)C(=O)N1C[C@@H]2C[C@H]1CN2C(=O)CNS(=O)(=O)c1cc(Cl)ccc1Cl

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PYGL P06737 7/20 0.41
CYP51A1 Q16850 7/20 0.41
PYGM P11217 1/20 0.41
SMYD3 Q9H7B4 2/20 0.38
LGALS8 O00214 2/20 0.38
BCAT1 P54687 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
LGALS3 P17931 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4056416 0.93 SMYD3 (0.39) PYGLCYP51A1PYGMSMYD3LGALS8
SCHEMBL4057673 0.91 PYGL (0.39) PYGLCYP51A1BCAT1
SCHEMBL4051117 0.91 ALOX15 (0.42) PYGLCYP51A1PYGMSMYD3LGALS8
SCHEMBL4049959 0.89 SMYD3 (0.41) PYGLCYP51A1PYGMSMYD3LGALS8
SCHEMBL4058202 0.88 ALB (0.38) CYP51A1
SCHEMBL4048476 0.87 PYGL (0.41) PYGLCYP51A1PYGMSMYD3MEN1
SCHEMBL8006223 0.86 PYGL (0.39) PYGLCYP51A1PYGMSMYD3LGALS8
SCHEMBL4056947 0.85 CCR1 (0.35) PYGLCYP51A1BCAT1
SCHEMBL4057362 0.85 PYGL (0.39) PYGLCYP51A1LGALS8BCAT1LGALS3
SCHEMBL4050168 0.84 DRD2 (0.36) PYGLCYP51A1PYGM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO claimed
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO disclosed