SCHEMBL4056416

SCHEMBL4056416

CC(C)(C)[C@H](NC(=O)c1cc2cc(F)ccc2[nH]1)C(=O)N1C[C@@H]2C[C@H]1CN2C(=O)CNS(=O)(=O)c1cc(C(F)(F)F)ccc1Cl

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.39
CYP51A1 Q16850 3/20 0.37
MCHR1 Q99705 1/20 0.37
PYGL P06737 3/20 0.36
PYGM P11217 2/20 0.36
LGALS8 O00214 1/20 0.36
LGALS3 P17931 1/20 0.36
ALDH1A1 P00352 1/20 0.34
PLD1 Q13393 1/20 0.34
MLLT1 Q03111 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
STAT6 P42226 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4052843 0.93 PYGL (0.41) SMYD3CYP51A1PYGLPYGMLGALS8
SCHEMBL4050168 0.92 DRD2 (0.36) CYP51A1MCHR1PYGLPYGMALDH1A1
SCHEMBL7983935 0.87 DRD2 (0.35) CYP51A1MCHR1PYGLPYGMALDH1A1
SCHEMBL7996360 0.86 SMYD3 (0.36) SMYD3CYP51A1MCHR1PYGLPYGM
SCHEMBL4059685 0.86 MCHR1 (0.39) SMYD3CYP51A1MCHR1PYGLPYGM
SCHEMBL4057673 0.83 PYGL (0.39) CYP51A1PYGLDRD2DRD3STAT6
SCHEMBL4051117 0.83 ALOX15 (0.42) SMYD3CYP51A1PYGLPYGMLGALS8
SCHEMBL4058360 0.83 DRD2 (0.36) CYP51A1MCHR1PYGLPYGMALDH1A1
SCHEMBL4049959 0.81 SMYD3 (0.41) SMYD3CYP51A1PYGLPYGMLGALS8
SCHEMBL4344872 0.81 SMYD3 (0.37) SMYD3CYP51A1MCHR1PYGLPYGM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO claimed
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO disclosed