SCHEMBL4056947

SCHEMBL4056947

Cc1cccc2[nH]c(C(=O)N[C@H](C(=O)N3C[C@@H]4C[C@H]3CN4C(=O)CNS(=O)(=O)c3cc(Cl)ccc3Cl)C(C)(C)C)cc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.35
BCAT1 P54687 2/20 0.33
PYGL P06737 2/20 0.32
DPP4 P27487 1/20 0.32
NR3C1 P04150 1/20 0.32
NPC1 O15118 1/20 0.31
CYP51A1 Q16850 2/20 0.31
MGAM O43451 1/20 0.31
GAA P10253 1/20 0.31
SI P14410 1/20 0.31
MGAM2 Q2M2H8 1/20 0.31
CASP1 P29466 1/20 0.31
CASP4 P49662 1/20 0.31
CASP5 P51878 1/20 0.31
CASP7 P55210 1/20 0.31
CASP9 P55211 1/20 0.31
CASP8 Q14790 1/20 0.31
CASP10 Q92851 1/20 0.31
EGFR P00533 1/20 0.31
NR1H2 P55055 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4058202 0.92 ALB (0.38) DPP4CYP51A1
SCHEMBL4057673 0.90 PYGL (0.39) BCAT1PYGLCYP51A1EGFR
SCHEMBL4051117 0.88 ALOX15 (0.42) BCAT1PYGLCYP51A1
SCHEMBL8007197 0.87 CCR1 (0.33) CCR1BCAT1PYGL
SCHEMBL4052843 0.85 PYGL (0.41) BCAT1PYGLCYP51A1
SCHEMBL4057362 0.84 PYGL (0.39) BCAT1PYGLCYP51A1EGFR
SCHEMBL4050168 0.82 DRD2 (0.36) PYGLCYP51A1
SCHEMBL4052196 0.82 DRD4 (0.38) PYGLCYP51A1EGFRNR1H2NR1H3
SCHEMBL4051255 0.82 CCR1 (0.41) CCR1DPP4CASP1CASP4CASP5
SCHEMBL4059459 0.80 PYGL (0.38) BCAT1PYGLCYP51A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO claimed
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO disclosed