SCHEMBL4057673

SCHEMBL4057673

CC(C)(C)[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@@H]2C[C@H]1CN2C(=O)CNS(=O)(=O)c1cc(Cl)ccc1Cl

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PYGL P06737 3/20 0.39
BCAT1 P54687 2/20 0.38
DRD2 P14416 1/20 0.38
CYP51A1 Q16850 5/20 0.37
EGFR P00533 1/20 0.36
DRD3 P35462 2/20 0.36
ALOX15 P16050 1/20 0.35
STAT6 P42226 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4057362 0.94 PYGL (0.39) PYGLBCAT1DRD2CYP51A1EGFR
SCHEMBL4051117 0.94 ALOX15 (0.42) PYGLBCAT1CYP51A1ALOX15
SCHEMBL4052196 0.92 DRD4 (0.38) PYGLDRD2CYP51A1EGFRDRD3
SCHEMBL4050168 0.92 DRD2 (0.36) PYGLDRD2CYP51A1DRD3STAT6
SCHEMBL4052843 0.91 PYGL (0.41) PYGLBCAT1CYP51A1
SCHEMBL4056947 0.90 CCR1 (0.35) PYGLBCAT1CYP51A1EGFR
SCHEMBL4059459 0.90 PYGL (0.38) PYGLBCAT1DRD2CYP51A1DRD3
SCHEMBL4058202 0.89 ALB (0.38) CYP51A1
SCHEMBL7993594 0.88 PYGL (0.40) PYGLBCAT1DRD2CYP51A1EGFR
SCHEMBL4056168 0.87 ALDH1A1 (0.42) PYGLBCAT1DRD2CYP51A1STAT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO claimed
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO disclosed