SCHEMBL4057362

SCHEMBL4057362

CC(C)(C)[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@@H]2C[C@H]1CN2C(=O)CNS(=O)(=O)c1ccc(Cl)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PYGL P06737 2/20 0.39
BCAT1 P54687 2/20 0.38
DRD2 P14416 1/20 0.38
CYP51A1 Q16850 5/20 0.37
LGALS8 O00214 3/20 0.37
LGALS1 P09382 1/20 0.37
LGALS3 P17931 1/20 0.37
DRD3 P35462 2/20 0.37
EGFR P00533 1/20 0.36
ALOX15 P16050 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4057673 0.94 PYGL (0.39) PYGLBCAT1DRD2CYP51A1DRD3
SCHEMBL4052196 0.90 DRD4 (0.38) PYGLDRD2CYP51A1DRD3EGFR
SCHEMBL4051527 0.90 DRD3 (0.39) PYGLBCAT1DRD2CYP51A1LGALS8
SCHEMBL4056496 0.89 TAS1R3 (0.46) PYGLCYP51A1DRD3
SCHEMBL4051117 0.88 ALOX15 (0.42) PYGLBCAT1CYP51A1LGALS8ALOX15
SCHEMBL4050168 0.87 DRD2 (0.36) PYGLDRD2CYP51A1DRD3
SCHEMBL4049330 0.87 PYGL (0.38) PYGLDRD2CYP51A1DRD3ALOX15
SCHEMBL4050835 0.86 DRD2 (0.39) PYGLDRD2CYP51A1
SCHEMBL4049377 0.86 CYP51A1 (0.39) PYGLDRD2CYP51A1DRD3
SCHEMBL4052843 0.85 PYGL (0.41) PYGLBCAT1CYP51A1LGALS8LGALS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO claimed
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO disclosed