SCHEMBL7983935

SCHEMBL7983935

CC(C)(S)[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@@H]2C[C@H]1CN2C(=O)CNS(=O)(=O)c1cc(C(F)(F)F)ccc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.35
HTR2C P28335 2/20 0.35
DRD3 P35462 2/20 0.35
MCHR1 Q99705 1/20 0.35
DRD1 P21728 1/20 0.35
DRD4 P21917 1/20 0.35
DRD5 P21918 1/20 0.35
CYP51A1 Q16850 2/20 0.35
ALDH1A1 P00352 1/20 0.34
HTR1A P08908 1/20 0.34
HTR2A P28223 1/20 0.34
PYGL P06737 1/20 0.33
PYGM P11217 1/20 0.33
CCKBR P32239 1/20 0.33
CTNNB1 P35222 1/20 0.32
ESR1 P03372 1/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
BCAT1 P54687 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050168 0.95 DRD2 (0.36) DRD2HTR2CDRD3MCHR1DRD1
SCHEMBL4056416 0.87 SMYD3 (0.39) DRD2DRD3MCHR1CYP51A1ALDH1A1
SCHEMBL4057673 0.86 PYGL (0.39) DRD2DRD3CYP51A1PYGLBCAT1
SCHEMBL4058360 0.85 DRD2 (0.36) DRD2HTR2CDRD3MCHR1DRD1
SCHEMBL4055536 0.83 DRD2 (0.35) DRD2HTR2CDRD3MCHR1DRD1
SCHEMBL4057362 0.82 PYGL (0.39) DRD2DRD3CYP51A1PYGLBCAT1
SCHEMBL19856858 0.82 DRD2 (0.39) DRD2HTR2CDRD3MCHR1DRD1
SCHEMBL19856857 0.82 DRD2 (0.39) DRD2HTR2CDRD3MCHR1DRD1
SCHEMBL7995568 0.81 DRD2 (0.34) DRD2HTR2CDRD3MCHR1DRD1
SCHEMBL4051117 0.80 ALOX15 (0.42) CYP51A1PYGLPYGMBCAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009146177-A1 TRPV4 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2009-12-03 WO disclosed