SCHEMBL4078455

SCHEMBL4078455

O=c1[nH]c2ccccc2cc1C1=CCNC(Cc2ccccc2)C1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.44
CHEK1 O14757 2/20 0.44
CDK5 Q00535 8/20 0.40
CDK5R1 Q15078 8/20 0.40
PDGFRB P09619 1/20 0.40
FGFR1 P11362 1/20 0.40
BRD4 O60885 1/20 0.37
DAO P14920 1/20 0.37
DDO Q99489 1/20 0.37
KDM4E B2RXH2 1/20 0.37
IL4I1 Q96RQ9 1/20 0.36
HDAC8 Q9BY41 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8368017 0.75 SLC6A3 (0.37) KDM4E
SCHEMBL5265951 0.72 POLB (0.44)
SCHEMBL7560334 0.72 POLB (0.39)
SCHEMBL5164934 0.71 HTR2A (0.34)
SCHEMBL9051187 0.70 CHRM2 (0.38) BRD4
SCHEMBL6504166 0.69 POLB (0.34)
SCHEMBL7844747 0.69 CDK9 (0.35)
SCHEMBL8312119 0.68 POLB (0.40)
SCHEMBL6683579 0.68 POLB (0.37)
SCHEMBL1813854 0.67 KDR (0.60) KDRCHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009020470-A2 CGRP RECEPTOR ANTAGONISTS VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-02-12 WO disclosed