SCHEMBL4078720

SCHEMBL4078720

Cc1occc1C(=O)Nc1n[nH]c2cc(C(=O)O)oc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 7/20 0.46
NPC1 O15118 7/20 0.46
RAB9A P51151 7/20 0.46
HTT P42858 5/20 0.46
ALDH1A1 P00352 6/20 0.45
PKM P14618 5/20 0.45
HPGD P15428 4/20 0.45
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.45
MAPK1 P28482 1/20 0.44
ESR2 Q92731 1/20 0.44
POLB P06746 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HSD17B10 Q99714 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
TSHR P16473 1/20 0.42
USP2 O75604 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4083487 0.84 SMN1; SMN2 (0.41) SMN1; SMN2NPC1RAB9AHTTALDH1A1
SCHEMBL4081816 0.84 MAPT (0.47) SMN1; SMN2NPC1RAB9AALDH1A1PKM
SCHEMBL2904998 0.81 GPR35 (0.47) SMN1; SMN2NPC1RAB9AALDH1A1HPGD
SCHEMBL4088557 0.80 SMN1; SMN2 (0.48) SMN1; SMN2NPC1RAB9AHTTALDH1A1
SCHEMBL4087457 0.80 KLK7 (0.47) SMN1; SMN2NPC1RAB9AHTTALDH1A1
SCHEMBL4086303 0.80 MAPK1 (0.49) SMN1; SMN2NPC1RAB9AALDH1A1PKM
SCHEMBL4078618 0.79 CDK7 (0.35) SMN1; SMN2NPC1RAB9AHTTPKM
SCHEMBL2913699 0.79 GPR35 (0.51) NPC1RAB9AHTTALDH1A1PKM
SCHEMBL2912045 0.78 CYP1A2 (0.42) HTTALDH1A1HPGDMAPK1CYP2C9
SCHEMBL4083540 0.78 FGFR1 (0.50) NPC1RAB9AHTTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058315-A1 1H-Furo[3,2-C]Pyrazoles active as aurora kinase inhibitors Nerviano Medical Sciences S.r.l. (IT) 2009-05-13 EP claimed
EP-2058315-A1 1H-Furo[3,2-C]Pyrazoles active as aurora kinase inhibitors Nerviano Medical Sciences S.r.l. (IT) 2009-05-13 EP disclosed