SCHEMBL4119682

SCHEMBL4119682

[CH2]OC(=O)NC(=O)C(Cl)(Cl)Cl

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 1/20 0.30
TP53 P04637 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4119686 0.77 L3MBTL1 (0.46) L3MBTL1ALDH1A1TP53TSHR
SCHEMBL712181 0.74 ALDH1A1 (0.44) L3MBTL1ALDH1A1TP53TSHR
SCHEMBL6955782 0.71 L3MBTL1 (0.33) L3MBTL1
SCHEMBL19500078 0.71 L3MBTL1 (0.38) L3MBTL1
SCHEMBL10360055 0.70 ALDH1A1 (0.41) L3MBTL1ALDH1A1
SCHEMBL19508784 0.70 HTT (0.41) L3MBTL1TSHR
SCHEMBL31734135 0.69 ALDH1A1 (0.39) L3MBTL1ALDH1A1TP53TSHR
SCHEMBL3136565 0.67 ALDH1A1 (0.44) L3MBTL1ALDH1A1TP53TSHR
SCHEMBL6969487 0.67 ALDH1A1 (0.37) L3MBTL1ALDH1A1TP53TSHR
SCHEMBL6959890 0.67 L3MBTL1 (0.32) L3MBTL1ALDH1A1TP53TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090004140-A1 4-SUBSTITUTED PYRROLIDINE AS ANTI-INFECTIVES ENANTA PHARMACEUTICALS, INC. 2009-01-01 US claimed
WO-2009003009-A1 SUBSTITUTED PYRROLIDINE AS ANTI-INFECTIVES ENANTA PHARMACEUTICALS, INC. (US) 2008-12-31 WO claimed
US-20090004140-A1 4-SUBSTITUTED PYRROLIDINE AS ANTI-INFECTIVES ENANTA PHARMACEUTICALS, INC. 2009-01-01 US disclosed
WO-2009003009-A1 SUBSTITUTED PYRROLIDINE AS ANTI-INFECTIVES ENANTA PHARMACEUTICALS, INC. (US) 2008-12-31 WO disclosed
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed
US-4729991-A SUBSTITUTED BY HETEROCYCLIC THIOMETHYL GROUP FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1988-03-08 US disclosed
US-4703046-A Cephem compounds and processes for preparation thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1987-10-27 US disclosed
US-4216215-A 7[(Furanyl-2-acetamido)-2-acetamido]cephalosporin derivatives PFIZER INC. (US) 1980-08-05 US disclosed
US-4137312-A Epoxy substituted cephalosporin derivatives PFIZER INC. (US) 1979-01-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090004140-A1 4-SUBSTITUTED PYRROLIDINE AS ANTI-INFECTIVES EIF2AK2, RNGTT, POLR2E L3MBTL1 2522/4885ALDH1A1 539/4885TP53 1967/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.