SCHEMBL4137813

SCHEMBL4137813

CCOC(=O)CCN(Cc1ccccc1)C(=O)OC(C)(C)C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC2 Q92769 1/20 0.51
NCOR2 Q9Y618 1/20 0.51
ALOX5 P09917 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
ALDH1A1 P00352 5/20 0.48
LTA4H P09960 2/20 0.46
CTSL P07711 1/20 0.46
CTSB P07858 1/20 0.46
CTSS P25774 1/20 0.46
LMNA P02545 3/20 0.45
HSD17B10 Q99714 2/20 0.45
POLB P06746 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
AKT1 P31749 2/20 0.44
NPC1 O15118 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1052780 0.87 HDAC3 (0.53) HDAC3HDAC1HDAC2NCOR2SMN1; SMN2
SCHEMBL5884593 0.87 HDAC1 (0.53) HDAC3HDAC1HDAC2NCOR2ALDH1A1
SCHEMBL3914953 0.85 ALOX5 (0.46) HDAC3HDAC1HDAC2NCOR2ALOX5
SCHEMBL4147838 0.85 HDAC1 (0.56) HDAC3HDAC1HDAC2NCOR2ALDH1A1
SCHEMBL9060170 0.84 HDAC1 (0.60) HDAC3HDAC1HDAC2NCOR2ALDH1A1
SCHEMBL17686967 0.82 SLC6A2 (0.48) SMN1; SMN2ALDH1A1LMNAPOLB
SCHEMBL20347975 0.81 REN (0.58) HDAC3HDAC1HDAC2ALOX5SMN1; SMN2
SCHEMBL2224578 0.81 SMN1; SMN2 (0.54) ALOX5SMN1; SMN2ALDH1A1LTA4HLMNA
SCHEMBL11728356 0.81 ALOX5 (0.48) ALOX5SMN1; SMN2ALDH1A1LTA4HLMNA
SCHEMBL3328177 0.81 HDAC3 (0.54) HDAC3HDAC1HDAC2NCOR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090182010-A1 COMPOUNDS HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY THERAVANCE BIOPHARMA R&D IP, LLC 2009-07-16 US disclosed
US-7528253-B2 Compounds having β2 adrenergic receptor agonist and muscarinic receptor antagonist activity THERAVANCE, INC. (US) 2009-05-05 US disclosed
US-20090062342-A1 AMINES ACTELION PHARMACEUTICALS LTD. (CH) 2009-03-05 US disclosed
US-20060116398-A1 Compounds having beta2 adrenergic receptor agonist and muscarinic receptor antagonist activity THERAVANCE BIOPHARMA R&D IP, LLC 2006-06-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090182010-A1 COMPOUNDS HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY ADRB2, ADRA2B, ADRA2A HDAC3 1584/4885HDAC1 1705/4885HDAC2 1119/4885
US-20090062342-A1 AMINES REN, ACE, MAOA HDAC3 3308/4885HDAC1 2808/4885HDAC2 1943/4885
US-20060116398-A1 Compounds having beta2 adrenergic receptor agonist and muscarinic receptor antagonist activity ADRB2, ADRA2B, ADRB1 HDAC3 1648/4885HDAC1 1770/4885HDAC2 1161/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.