SCHEMBL4154967

SCHEMBL4154967

O=C(O)c1cc2cc(Cl)cc(F)c2[nH]1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 6/20 0.59
F7 P08709 1/20 0.51
F3 P13726 1/20 0.51
PYGL P06737 2/20 0.46
IDO1 P14902 2/20 0.46
TDO2 P48775 2/20 0.46
EIF4A3 P38919 3/20 0.44
ALDH1A1 P00352 3/20 0.44
HPGD P15428 3/20 0.44
KDM4E B2RXH2 2/20 0.44
LMNA P02545 2/20 0.44
HSD17B10 Q99714 2/20 0.44
GRIN1 Q05586 1/20 0.44
PDPK1 O15530 1/20 0.44
TSHR P16473 1/20 0.44
NFKB1 P19838 1/20 0.44
APEX1 P27695 1/20 0.44
CYP2C19 P33261 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
PYGM P11217 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2576853 0.84 HPGD (0.56) HRH4F7F3IDO1TDO2
SCHEMBL3274871 0.82 HRH4 (0.56) HRH4F7F3ALDH1A1HPGD
SCHEMBL16235908 0.81 HRH4 (0.56) HRH4PYGLPYGM
SCHEMBL17865579 0.79 HRH4 (0.58) HRH4F7F3ALDH1A1HPGD
SCHEMBL22396281 0.79 HRH4 (0.59) HRH4F7F3ALDH1A1HPGD
SCHEMBL25531648 0.79 PIN1 (0.51) HRH4IDO1TDO2EIF4A3ALDH1A1
SCHEMBL18661924 0.79 IDO1 (0.46) HRH4IDO1TDO2EIF4A3ALDH1A1
SCHEMBL21225606 0.78 EIF4A3 (0.50) HRH4F7F3IDO1TDO2
SCHEMBL8959651 0.78 EIF4A3 (0.54) F7F3IDO1TDO2EIF4A3
SCHEMBL16486363 0.77 ALOX15 (0.56) HRH4PYGLALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12018033-B2 Inhibitors of protein arginine deiminases FORWARD THERAPEUTICS, INC. (US) 2024-06-25 US disclosed
US-20230151018-A1 INHIBITORS OF PROTEIN ARGININE DEIMINASES FORWARD THERAPEUTICS, INC. 2023-05-18 US disclosed
US-20230151018-A1 INHIBITORS OF PROTEIN ARGININE DEIMINASES FORWARD THERAPEUTICS, INC. 2023-05-18 US disclosed
US-20230151018-A1 INHIBITORS OF PROTEIN ARGININE DEIMINASES FORWARD THERAPEUTICS, INC. 2023-05-18 US disclosed
US-11453676-B2 Inhibitors of protein arginine deiminases FORWARD THERAPEUTICS, INC. (US) 2022-09-27 US disclosed
US-20210053975-A1 INHIBITORS OF PROTEIN ARGININE DEIMINASES FORWARD THERAPEUTICS, INC. 2021-02-25 US disclosed
US-20210053975-A1 INHIBITORS OF PROTEIN ARGININE DEIMINASES FORWARD THERAPEUTICS, INC. 2021-02-25 US disclosed
EP-3746430-A1 INHIBITORS OF PROTEIN ARGININE DEIMINASES Padforward LLC (US) 2020-12-09 EP disclosed
WO-2019152883-A1 INHIBITORS OF PROTEIN ARGININE DEIMINASES PADFORWARD LLC (US) 2019-08-08 WO disclosed
US-20090124682-A1 Indan-Amide Derivatives with Glycogen Phosphorylase Inhibitory Activity BIRCH ALAN MARTIN 2009-05-14 US disclosed
US-20090124682-A1 Indan-Amide Derivatives with Glycogen Phosphorylase Inhibitory Activity BIRCH ALAN MARTIN 2009-05-14 US disclosed
US-20090124682-A1 Indan-Amide Derivatives with Glycogen Phosphorylase Inhibitory Activity BIRCH ALAN MARTIN 2009-05-14 US disclosed
EP-1848693-A1 INDAN-AMIDE DERIVATIVES WITH GLYCOGEN PHOSPHORYLASE INHIBITORY ACTIVITY AstraZeneca AB (SE) 2007-10-31 EP disclosed
WO-2006082400-A1 INDAN-AMIDE DERIVATIVES WITH GLYCOGEN PHOSPHORYLASE INHIBITORY ACTIVITY ASTRAZENECA AB (SE) 2006-08-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230151018-A1 INHIBITORS OF PROTEIN ARGININE DEIMINASES PADI2, PADI1, PADI4 HRH4 2377/4885F7 4510/4885F3 3103/4885
US-11453676-B2 Inhibitors of protein arginine deiminases PADI2, PADI1, PADI4 HRH4 2617/4885F7 4529/4885F3 2476/4885
US-20090124682-A1 Indan-Amide Derivatives with Glycogen Phosphorylase Inhibitory Activity PYGL, PYGM, GYS1 HRH4 4670/4885F7 4226/4885F3 3479/4885
US-20210053975-A1 INHIBITORS OF PROTEIN ARGININE DEIMINASES PADI2, PADI1, PADI4 HRH4 2377/4885F7 4510/4885F3 3103/4885
US-12018033-B2 Inhibitors of protein arginine deiminases PADI2, PADI1, PADI4 HRH4 2369/4885F7 4400/4885F3 2061/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.