SCHEMBL4177982

SCHEMBL4177982

COc1ccc2c(Cl)cc(-c3c[nH]nc3CCN3CCOCC3)nc2c1C

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.40
KDM4E B2RXH2 2/20 0.38
LMNA P02545 2/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
ATM Q13315 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TNIK Q9UKE5 1/20 0.38
BRD4 O60885 1/20 0.37
CREBBP Q92793 1/20 0.37
PDPK1 O15530 1/20 0.37
SUV39H2 Q9H5I1 1/20 0.37
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
TP53 P04637 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4187144 0.89 ALDH1A1 (0.38) ACHEKDM4ELMNAALDH1A1MAPT
SCHEMBL4189834 0.83 MAPK1 (0.37) KDM4ELMNAALDH1A1MAPTNPSR1
SCHEMBL4185269 0.81 KDM4E (0.34) KDM4EALDH1A1MAPTHSD17B10PDPK1
SCHEMBL4177972 0.80 SLC10A2 (0.33) KDM4EHSP90AA1HSP90AB1
SCHEMBL4177980 0.78 S1PR1 (0.48) KDM4ELMNAALDH1A1MAPTATM
SCHEMBL4177976 0.78 KMT2A (0.31) KDM4EPDPK1
SCHEMBL4182671 0.76 KDR (0.35) KDM4EALDH1A1MAPTBRD4HSP90AA1
SCHEMBL4178311 0.71 PDE10A (0.35) KDM4EALDH1A1MAPTHSD17B10
SCHEMBL4191730 0.69 SLC10A2 (0.33) ALDH1A1MAPT
SCHEMBL4182845 0.69 MAPT (0.34) KDM4ELMNAALDH1A1MAPTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009014730-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS, INC. (US) 2009-01-29 WO disclosed