SCHEMBL4177972

SCHEMBL4177972

COc1ccc2c(Cl)cc(-c3c[nH]nc3CCC(C)C)nc2c1C

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC10A2 Q12908 1/20 0.33
AAK1 Q2M2I8 2/20 0.32
KMT2A Q03164 1/20 0.30
PDE4D Q08499 1/20 0.30
RAD52 P43351 1/20 0.30
HSP90AA1 P07900 1/20 0.30
HSP90AB1 P08238 1/20 0.30
KDM4E B2RXH2 1/20 0.30
GAA P10253 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4177976 0.90 KMT2A (0.31) KMT2APDE4DRAD52KDM4EGAA
SCHEMBL4189834 0.89 MAPK1 (0.37) KMT2APDE4DRAD52KDM4EHTT
SCHEMBL4191730 0.88 SLC10A2 (0.33) SLC10A2AAK1KMT2APDE4DRAD52
SCHEMBL4185269 0.86 KDM4E (0.34) KMT2APDE4DRAD52KDM4EHTT
SCHEMBL4182671 0.82 KDR (0.35) KMT2APDE4DHSP90AA1HSP90AB1KDM4E
SCHEMBL4177982 0.80 ACHE (0.40) HSP90AA1HSP90AB1KDM4E
SCHEMBL4183205 0.77 KDM4E (0.33) KMT2ARAD52KDM4EGAA
SCHEMBL4178311 0.76 PDE10A (0.35) KMT2ARAD52KDM4EGAAHTT
SCHEMBL4182845 0.73 MAPT (0.34) SLC10A2KMT2APDE4DRAD52KDM4E
SCHEMBL4177971 0.73 PRMT5 (0.39) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009014730-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS, INC. (US) 2009-01-29 WO disclosed