SCHEMBL4188150

SCHEMBL4188150

C=CS(=O)(=O)c1ccc(OC)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.70
RAB9A P51151 2/20 0.70
ALDH1A1 P00352 2/20 0.70
LMNA P02545 1/20 0.70
TP53 P04637 1/20 0.70
MAPT P10636 1/20 0.70
TSHR P16473 1/20 0.70
XBP1 P17861 1/20 0.70
MAPK1 P28482 1/20 0.70
HTT P42858 1/20 0.70
MDM2 Q00987 1/20 0.70
SMN1; SMN2 Q16637 1/20 0.70
HSD17B10 Q99714 1/20 0.70
PKM P14618 4/20 0.59
NFE2L2 Q16236 5/20 0.51
CA1 P00915 3/20 0.50
CA2 P00918 3/20 0.50
MMP1 P03956 1/20 0.50
MMP2 P08253 1/20 0.50
MMP9 P14780 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10860893 0.82 ALDH1A1 (0.73) NPC1RAB9AALDH1A1LMNATP53
SCHEMBL7379397 0.81 PKM (0.61) NPC1RAB9AALDH1A1HTTPKM
SCHEMBL7034773 0.79 ALDH1A1 (0.63) NPC1RAB9AALDH1A1LMNATP53
SCHEMBL2872244 0.79 PKM (0.53) NPC1RAB9AALDH1A1LMNATP53
SCHEMBL11340502 0.79 LMNA (0.63) NPC1RAB9AALDH1A1LMNATP53
SCHEMBL8684013 0.77 NFE2L2 (0.56) NPC1RAB9AALDH1A1LMNATP53
Ethylene SCHEMBL28422227 0.77 PKM (0.61) NPC1RAB9AALDH1A1LMNAHTT
SCHEMBL31653833 0.76 ALDH1A1 (0.66) NPC1RAB9AALDH1A1LMNATP53
SCHEMBL26618987 0.76 ALDH1A1 (0.66) NPC1RAB9AALDH1A1LMNATP53
SCHEMBL27494242 0.76 PKM (0.55) NPC1RAB9AALDH1A1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118184684-A Method for preparing beta-sulfonyl borate in water/organic two-phase 成都理工大学 2024-06-14 CN claimed
CN-118184684-A Method for preparing beta-sulfonyl borate in water/organic two-phase 成都理工大学 2024-06-14 CN disclosed
US-10882029-B1 Graphene oxide and cobalt tin oxide nanocomposite and method of use KING FAHD UNIVERSITY OF PETROLEUM AND MINERALS (SA) 2021-01-05 US disclosed
US-9353142-B2 Protecting group for indole group, nucleic acid-synthesizing amidite and nucleic acid-synthesizing method APTA BIOSCIENCES LTD. (GB) 2016-05-31 US disclosed
US-20140256928-A1 PROTECTING GROUP FOR INDOLE GROUP, NUCLEIC ACID-SYNTHESIZING AMIDITE AND NUCLEIC ACID-SYNTHESIZING METHOD APTA BIOSCIENCES LTD. (GB) 2014-09-11 US disclosed
US-20090247536-A1 Bissulfonamide Compounds As Agonists Of GalR1, Compositions, And Methods Of Use MJALLI ADNAN M M 2009-10-01 US disclosed
US-7582673-B2 Benzo[b]thiophene-2-sulfonic acid [2-(2-chloro-5-trifluoromethylbenzenesulfonylamino)phenyl] amide; agonists of GalR1; useful in treating neuropathic pain or cancer HIGH POINT PHARMACEUTICALS, LLC (US) 2009-09-01 US disclosed
EP-1809619-A1 BISSULFONAMIDE COMPOUNDS AS AGONISTS OF GALR1, COMPOSITIONS, AND METHODS OF USE Transtech Pharma, Inc. (US) 2007-07-25 EP disclosed
US-20060106089-A1 Bissulfonamide compounds as agonists of GalR1, compositions, and methods of use VTVX HOLDINGS II LLC 2006-05-18 US disclosed
WO-2006047302-A1 BISSULFONAMIDE COMPOUNDS AS AGONISTS OF GALR1, COMPOSITIONS, AND METHODS OF USE TRANSTECH PHARMA, INC. (US) 2006-05-04 WO disclosed
EP-0841323-B1 Method for producing arylvinylsulfone SUMITOMO CHEMICAL CO (JP) 2003-03-05 EP disclosed
US-5902905-A Method for producing arylvinylsulfone SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-05-11 US disclosed
EP-0841323-A2 Method for producing arylvinylsulfone SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1998-05-13 EP disclosed
US-4260552-A INSECTICIDES, HERBICIDES UNIROYAL, INC. (US) 1981-04-07 US disclosed
US-4160846-A Method for controlling insects with tetrasubstituted organotin compounds UNIROYAL, INC. (US) 1979-07-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140256928-A1 PROTECTING GROUP FOR INDOLE GROUP, NUCLEIC ACID-SYNTHESIZING AMIDITE AND NUCLEIC ACID-SYNTHESIZING METHOD INMT, NSUN2, RNMT NPC1 2034/4885RAB9A 4068/4885ALDH1A1 2229/4885
US-20060106089-A1 Bissulfonamide compounds as agonists of GalR1, compositions, and methods of use GALR1, GALR3, GALR2 NPC1 4565/4885RAB9A 2045/4885ALDH1A1 4001/4885
US-20090247536-A1 Bissulfonamide Compounds As Agonists Of GalR1, Compositions, And Methods Of Use GALR1, GALR3, GALR2 NPC1 4565/4885RAB9A 2045/4885ALDH1A1 4001/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.