SCHEMBL4204113

SCHEMBL4204113

NC(=O)C(C1CCCCC1)(C1CCCCC1)N(CC(=O)O)C(=O)C(=O)c1c[nH]c2cc(CO)ccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PRKAB2 O43741 2/20 0.33
PRKAG1 P54619 2/20 0.33
PRKAA2 P54646 2/20 0.33
PRKAA1 Q13131 2/20 0.33
PRKAG3 Q9UGI9 2/20 0.33
PRKAG2 Q9UGJ0 2/20 0.33
PRKAB1 Q9Y478 2/20 0.33
RAB9A P51151 2/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
NPC1 O15118 1/20 0.33
GABRA1 P14867 6/20 0.33
GABRB2 P47870 6/20 0.33
GABRG2 P18507 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3950315 0.87 ALDH1A1 (0.39) ALDH1A1MAPTL3MBTL1RAB9AHTR3E
SCHEMBL4029168 0.81 ALDH1A1 (0.51) ALDH1A1MAPTL3MBTL1NPC1
SCHEMBL4025964 0.80 ALDH1A1 (0.51) ALDH1A1MAPTL3MBTL1NPC1
SCHEMBL4029459 0.80 CCR5 (0.42) ALDH1A1RAB9ANPC1GABRA1GABRB2
SCHEMBL3939700 0.76 ALDH1A1 (0.42) ALDH1A1MAPTL3MBTL1PRKAB2PRKAG1
SCHEMBL4199729 0.76 ALDH1A1 (0.41) ALDH1A1MAPTL3MBTL1RAB9ANPC1
SCHEMBL3939702 0.73 RAB9A (0.42) ALDH1A1MAPTL3MBTL1RAB9ANPC1
SCHEMBL4204118 0.71 HDAC1 (0.35) ALDH1A1MAPTL3MBTL1PRKAB2PRKAG1
SCHEMBL4023062 0.70 MAPT (0.38) ALDH1A1MAPTL3MBTL1
SCHEMBL1558428 0.69 PRKAB2 (0.50) MAPTPRKAB2PRKAG1PRKAA2PRKAA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009019508-A1 CALCIUM ION CHANNEL MODULATORS & USES THEREOF LECTUS THERAPEUTICS LIMITED (GB) 2009-02-12 WO disclosed