Apocynin

Apocynin

SCHEMBL4232138

COc1cc(C(C)=O)ccc1O.Oc1ccccc1

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.65
SLC22A6 Q4U2R8 1/20 0.62
SLC22A8 Q8TCC7 1/20 0.62
MEN1 O00255 1/20 0.62
RAB9A P51151 1/20 0.62
KMT2A Q03164 1/20 0.62
HSD17B2 P37059 1/20 0.53
LMNA P02545 1/20 0.51
CYP1A2 P05177 1/20 0.51
HSP90AA1 P07900 1/20 0.51
HSP90AB1 P08238 1/20 0.51
BLM P54132 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
AKR1C3 P42330 1/20 0.51
AKR1C2 P52895 1/20 0.51
GAA P10253 1/20 0.51
MAOB P27338 1/20 0.50
KDM4E B2RXH2 1/20 0.50
POLB P06746 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Apocynin SCHEMBL109372 0.90 HTT (0.73) HTTSLC22A6SLC22A8MEN1RAB9A
Apocynin SCHEMBL108512 0.90 HTT (0.73) HTTSLC22A6SLC22A8MEN1RAB9A
Apocynin SCHEMBL28429584 0.90 HTT (0.73) HTTSLC22A6SLC22A8MEN1RAB9A
Apocynin SCHEMBL109514 0.90 MEN1 (0.75) HTTSLC22A6SLC22A8MEN1RAB9A
Apocynin SCHEMBL29364797 0.90 MEN1 (0.75) HTTSLC22A6SLC22A8MEN1RAB9A
Apocynin SCHEMBL464770 0.90 MEN1 (0.75) HTTSLC22A6SLC22A8MEN1RAB9A
Vanillic Acid SCHEMBL28312392 0.89 HTT (0.83) HTTSLC22A6SLC22A8MEN1RAB9A
Apocynin SCHEMBL1859599 0.89 SLC22A6 (0.64) HTTSLC22A6SLC22A8MEN1RAB9A
Apocynin SCHEMBL28537029 0.88 HTT (0.71) HTTSLC22A6SLC22A8MEN1RAB9A
Apocynin SCHEMBL30937977 0.88 MEN1 (0.72) HTTSLC22A6SLC22A8MEN1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024115926-A1 FORMULATION COMPRISING APOCYNIN AND PAEONOL AKL RESEARCH & DEVELOPMENT LTD (GB) 2024-06-06 WO disclosed
CN-116999417-A Liquid preparation containing paeonol and apocynin AKL研究发展有限公司 2023-11-07 CN disclosed
US-20230330017-A1 LIQUID FORMULATION COMPRISING PAEONOL AND APOCYNIN AKL RES & DEVELOPMENT LTD (GB) 2023-10-19 US disclosed
CN-111372572-B Liquid preparation containing paeonol and apocynin AKL研究发展有限公司 2023-08-29 CN disclosed
US-11701325-B2 Liquid formulation comprising paeonol and apocynin AKL RESEARCH & DEVELOPMENT LTD (GB) 2023-07-18 US disclosed
EP-4019005-A1 LIQUID FORMULATION COMPRISING PAEONOL AND APOCYNIN AKL Research&Development Ltd (GB) 2022-06-29 EP disclosed
US-20220089600-A1 TGFß INHIBITOR AND PRODRUGS FUNDACIÓ INSTITUT DE RECERCA BIOMÈDICA (IRB BARCELONA) (ES) 2022-03-24 US disclosed
EP-3713546-B1 LIQUID FORMULATION COMPRISING PAEONOL AND APOCYNIN AKL RESEARCH&DEVELOPMENT LTD (GB) 2021-12-08 EP disclosed
EP-3883556-A2 TGF? INHIBITOR AND PRODRUGS Fundació Institut de Recerca Biomèdica IRB (Barcelona) (ES) 2021-09-29 EP disclosed
EP-3713546-A1 LIQUID FORMULATION COMPRISING PAEONOL AND APOCYNIN AKL Research&Development Ltd (GB) 2020-09-30 EP disclosed
US-20200297628-A1 LIQUID FORMULATION COMPRISING PAEONOL AND APOCYNIN AKL RESEARCH & DEVELOPMENT LTD (GB) 2020-09-24 US disclosed
CN-111372572-A Liquid preparation containing paeonol and apocynin AKL研究发展有限公司 2020-07-03 CN disclosed
WO-2019101842-A1 LIQUID FORMULATION COMPRISING PAEONOL AND APOCYNIN AKL RESEARCH & DEVELOPMENT LTD (GB) 2019-05-31 WO disclosed
WO-2013037843-A1 FORMULATION FOR THE TREATMENT OF BENIGN PROSTATE HYPERPLASIA AKL INFLAMMATORY LIMITED (GB) 2013-03-21 WO disclosed
EP-1868586-B1 ANTI-INFLAMMATORY FORMULATION AKL INFLAMMATORY LTD (GB) 2012-11-21 EP disclosed
US-20090215886-A1 Anti-Inflammatory Formulation AKL RESEARCH AND DEVELOPMENT LIMITED (GB) 2009-08-27 US disclosed
EP-1868586-A1 ANTI-INFLAMMATORY FORMULATION AKL Inflammatory Limited (GB) 2007-12-26 EP disclosed
WO-2006106350-A1 ANTI-INFLAMMATORY FORMULATION AKL INFLAMMATORY LIMITED (GB) 2006-10-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11701325-B2 Liquid formulation comprising paeonol and apocynin LPL, PNLIP, LPO HTT 1028/4885SLC22A6 1497/4885SLC22A8 2830/4885
US-20220089600-A1 TGFß INHIBITOR AND PRODRUGS TGFB1, TGFBR1, TGFBR2 HTT 4458/4885SLC22A6 809/4885SLC22A8 1079/4885
US-20090215886-A1 Anti-Inflammatory Formulation IL1B, MPO, TNF HTT 1164/4885SLC22A6 2502/4885SLC22A8 3974/4885
US-20200297628-A1 LIQUID FORMULATION COMPRISING PAEONOL AND APOCYNIN LPL, PNLIP, LIPA HTT 1366/4885SLC22A6 1080/4885SLC22A8 2269/4885
US-20230330017-A1 LIQUID FORMULATION COMPRISING PAEONOL AND APOCYNIN LPL, PNLIP, LPO HTT 1028/4885SLC22A6 1497/4885SLC22A8 2830/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.