SCHEMBL4312756

SCHEMBL4312756

O=C(CN(CC1CCCCC1)C(=O)C(=O)c1c[nH]c2cc(F)ccc12)NC1CCCCC1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.47
HDAC6 Q9UBN7 5/20 0.47
ALDH1A1 P00352 4/20 0.46
KMT2A Q03164 1/20 0.46
RAB9A P51151 4/20 0.44
NPC1 O15118 3/20 0.44
TDO2 P48775 1/20 0.40
MAPT P10636 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.37
MITF O75030 1/20 0.37
LMNA P02545 1/20 0.37
PKM P14618 1/20 0.37
XBP1 P17861 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4306692 0.94 HDAC1 (0.42) HDAC1HDAC6ALDH1A1KMT2ARAB9A
SCHEMBL3120950 0.88 ALDH1A1 (0.40) ALDH1A1KMT2ARAB9ANPC1TDO2
SCHEMBL4304078 0.85 MAPK14 (0.43) HDAC1HDAC6ALDH1A1KMT2AMAPT
SCHEMBL7985731 0.85 MAPT (0.55) HDAC1HDAC6ALDH1A1KMT2ARAB9A
SCHEMBL4312470 0.84 ALDH1A1 (0.42) HDAC1HDAC6ALDH1A1KMT2AMAPT
SCHEMBL4308534 0.84 ADRA1D (0.43) ALDH1A1KDM4E
SCHEMBL4313368 0.83 ALDH1A1 (0.43) HDAC1HDAC6ALDH1A1RAB9ATDO2
SCHEMBL4310271 0.83 ALDH1A1 (0.41) ALDH1A1MAPTL3MBTL1ROCK2ROCK1
SCHEMBL4305038 0.82 MAPT (0.51) HDAC1HDAC6ALDH1A1KMT2ARAB9A
SCHEMBL3121013 0.82 ALDH1A1 (0.40) ALDH1A1KMT2AMAPTL3MBTL1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133387-A1 INDOLE- 3 -GLYOXYLAMIDE DERIVATIVES FOR USE AS CALCIUM ION CHANNEL MODULATORS LECTUS THERAPEUTICS LIMITED (GB) 2009-11-05 WO claimed
WO-2009133387-A1 INDOLE- 3 -GLYOXYLAMIDE DERIVATIVES FOR USE AS CALCIUM ION CHANNEL MODULATORS LECTUS THERAPEUTICS LIMITED (GB) 2009-11-05 WO disclosed