SCHEMBL3120950

SCHEMBL3120950

O=C(O)CN(CC1CCCCC1)C(=O)C(=O)c1c[nH]c2cc(F)ccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
MAPT P10636 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MAPK14 Q16539 2/20 0.39
KMT2A Q03164 1/20 0.39
PKM P14618 2/20 0.38
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38
TDO2 P48775 1/20 0.37
DRD2 P14416 1/20 0.37
HTR2A P28223 1/20 0.37
HTR7 P34969 1/20 0.37
KCNH2 Q12809 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SLC6A4 P31645 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRK1 P41145 1/20 0.36
OPRL1 P41146 1/20 0.36
ADRA1D P25100 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4304078 0.89 MAPK14 (0.43) ALDH1A1MAPTL3MBTL1MAPK14KMT2A
SCHEMBL4313368 0.88 ALDH1A1 (0.43) ALDH1A1MAPTL3MBTL1MAPK14TDO2
SCHEMBL4312756 0.88 HDAC1 (0.47) ALDH1A1MAPTL3MBTL1KMT2APKM
SCHEMBL4310271 0.87 ALDH1A1 (0.41) ALDH1A1MAPTL3MBTL1MAPK14ROCK2
SCHEMBL3121013 0.86 ALDH1A1 (0.40) ALDH1A1MAPTL3MBTL1MAPK14KMT2A
SCHEMBL3122360 0.85 ALDH1A1 (0.59) ALDH1A1MAPTL3MBTL1KMT2ANPC1
SCHEMBL4315207 0.85 ALDH1A1 (0.45) ALDH1A1MAPTL3MBTL1KMT2AROCK2
SCHEMBL3945339 0.84 ALDH1A1 (0.42) ALDH1A1MAPTL3MBTL1MAPK14KMT2A
SCHEMBL4306692 0.84 HDAC1 (0.42) ALDH1A1MAPTL3MBTL1KMT2AROCK2
SCHEMBL7982425 0.84 PKM (0.43) ALDH1A1MAPTL3MBTL1MAPK14KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010035032-A1 CALCIUM ION CHANNEL MODULATORS & USES THEREOF LECTUS THERAPEUTICS LIMITED (GB) 2010-04-01 WO disclosed
WO-2010035032-A1 CALCIUM ION CHANNEL MODULATORS & USES THEREOF LECTUS THERAPEUTICS LIMITED (GB) 2010-04-01 WO disclosed
WO-2009133387-A1 INDOLE- 3 -GLYOXYLAMIDE DERIVATIVES FOR USE AS CALCIUM ION CHANNEL MODULATORS LECTUS THERAPEUTICS LIMITED (GB) 2009-11-05 WO disclosed
WO-2009133387-A1 INDOLE- 3 -GLYOXYLAMIDE DERIVATIVES FOR USE AS CALCIUM ION CHANNEL MODULATORS LECTUS THERAPEUTICS LIMITED (GB) 2009-11-05 WO disclosed