SCHEMBL4358364

SCHEMBL4358364

CNC(=O)OCc1nccs1

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 16/20 0.47
ALDH1A1 P00352 1/20 0.45
PKM P14618 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13264272 0.84 CYP3A4 (0.48) CYP3A4ALDH1A1PKML3MBTL1
SCHEMBL13234062 0.83 CYP3A4 (0.45) CYP3A4ALDH1A1PKML3MBTL1
SCHEMBL8316849 0.81 ALDH1A1 (0.46) CYP3A4ALDH1A1PKML3MBTL1
SCHEMBL16907555 0.78 NPC1 (0.60) CYP3A4ALDH1A1PKM
SCHEMBL19765222 0.78 CYP3A4 (0.46) CYP3A4ALDH1A1PKM
SCHEMBL20724252 0.78 ALDH1A1 (0.46) CYP3A4ALDH1A1PKML3MBTL1
SCHEMBL30845136 0.77 FDPS (0.42) CYP3A4ALDH1A1PKM
SCHEMBL7268929 0.77 CYP3A4 (0.51) CYP3A4
SCHEMBL7268924 0.77 CYP3A4 (0.51) CYP3A4
SCHEMBL3432947 0.77 L3MBTL1 (0.47) CYP3A4ALDH1A1PKML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8470863-B2 Derivatives and analogs of chroman as functionally selective ALPHA2C adrenoreceptor agonists MERCK SHARP & DOHME, CORP. (US) 2013-06-25 US disclosed
US-20100168195-A1 DERIVATIVES AND ANALOGS OF CHROMAN AS FUNCTIONALLY SELECTIVE ALPHA2C ADRENORECEPTOR AGONISTS MERCK SHARP & DOHME CORP. 2010-07-01 US disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100168195-A1 DERIVATIVES AND ANALOGS OF CHROMAN AS FUNCTIONALLY SELECTIVE ALPHA2C ADRENORECEPTOR AGONISTS ADRA2C, ADRB2, ADRA2A CYP3A4 1017/4885ALDH1A1 1551/4885PKM 2011/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.