SCHEMBL437559

SCHEMBL437559

Nc1c(Cl)cnc2c(OC(F)(F)F)cccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HAVCR2 Q8TDQ0 1/20 0.40
TNF P01375 1/20 0.38
LITAF Q99732 1/20 0.38
P2RX7 Q99572 1/20 0.37
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
HPGD P15428 1/20 0.36
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
MPL P40238 1/20 0.35
CTSC P53634 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
NR4A2 P43354 1/20 0.34
KDM4E B2RXH2 1/20 0.33
GRIA1 P42261 1/20 0.33
CACNG8 Q8WXS5 1/20 0.33
ACHE P22303 1/20 0.33
KMO O15229 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL437620 0.82 ALOX5AP (0.38) HAVCR2TNFLITAFADORA2AADORA1
SCHEMBL436008 0.80 HTR1A (0.44) HAVCR2CYP3A4KDM4E
SCHEMBL437574 0.77 PARP1 (0.45) HAVCR2NR4A2
SCHEMBL441707 0.76 HAVCR2 (0.63) HAVCR2CYP1A2NR4A2KDM4EACHE
SCHEMBL23497102 0.75 PDE4A (0.42) TNFLITAFP2RX7ADORA2AADORA1
SCHEMBL29828879 0.75 PI4KA (0.42) TNFLITAFADORA2AADORA1ALOX5AP
SCHEMBL29829215 0.75 PDE4A (0.42) TNFLITAFP2RX7ADORA2AADORA1
SCHEMBL441422 0.74 HAVCR2 (0.46) HAVCR2NR4A2ACHE
SCHEMBL29233308 0.73 TNF (0.39) TNFLITAFADORA2AADORA1ALOX5AP
SCHEMBL29989486 0.72 PIN1 (0.45) TNFLITAFHPGDKDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed