SCHEMBL435849

SCHEMBL435849

COc1cccc2c(N)c(Br)cnc12

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.44
ADRA1D P25100 2/20 0.44
ADRA1A P35348 2/20 0.44
ADRA1B P35368 2/20 0.44
EGFR P00533 1/20 0.44
HPGDS O60760 1/20 0.43
NSD2 O96028 1/20 0.43
CASP6 P55212 1/20 0.43
MCHR1 Q99705 1/20 0.42
ATP4A P20648 2/20 0.42
ATP4B P51164 2/20 0.42
CYP3A4 P08684 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
EP300 Q09472 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL436008 0.81 HTR1A (0.44) HTR1AADRA1DADRA1AADRA1BHPGDS
SCHEMBL437620 0.80 ALOX5AP (0.38) MCHR1
SCHEMBL442133 0.79 BACE1 (0.41) EGFR
SCHEMBL441701 0.78 ALDH1A1 (0.43) HTR1AADRA1DADRA1AADRA1BTDP1
SCHEMBL439862 0.76 HAVCR2 (0.63)
SCHEMBL436963 0.75 PDE5A (0.38) NSD2CASP6EP300
SCHEMBL435823 0.75 PARP1 (0.41) CYP3A4
SCHEMBL441951 0.75 HAVCR2 (0.58)
SCHEMBL4014412 0.75 HTR1A (0.59) HTR1AADRA1DADRA1AADRA1BEGFR
SCHEMBL30543156 0.75 HTR1A (0.59) HTR1AADRA1DADRA1AADRA1BEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed