SCHEMBL4366139

SCHEMBL4366139

CCCCOC(=O)n1cccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
BCHE P06276 1/20 0.47
TSHR P16473 7/20 0.47
L3MBTL1 Q9Y468 3/20 0.47
TDP1 Q9NUW8 2/20 0.47
LMNA P02545 4/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
POLB P06746 1/20 0.46
ATM Q13315 1/20 0.45
HPGD P15428 1/20 0.42
MAPK1 P28482 3/20 0.42
CYP3A4 P08684 3/20 0.42
TP53 P04637 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ESR1 P03372 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28810272 0.94 TSHR (0.49) ALDH1A1BCHETSHRL3MBTL1TDP1
SCHEMBL23953095 0.88 ALDH1A1 (0.44) ALDH1A1BCHETSHRL3MBTL1TDP1
SCHEMBL27810242 0.79 ALDH1A1 (0.42) ALDH1A1BCHETSHRL3MBTL1LMNA
SCHEMBL30403372 0.77 TSHR (0.53) ALDH1A1BCHETSHRL3MBTL1TDP1
SCHEMBL943943 0.77 SMN1; SMN2 (0.44) ALDH1A1BCHETSHRL3MBTL1TDP1
SCHEMBL28030479 0.75 ESR1 (0.49) ALDH1A1BCHETSHRL3MBTL1TDP1
SCHEMBL27295005 0.73 MEN1 (0.54) ALDH1A1TSHRL3MBTL1TDP1SMN1; SMN2
SCHEMBL4566478 0.73 NOS1 (0.46) ALDH1A1BCHETSHRL3MBTL1TDP1
SCHEMBL4780587 0.73 LMNA (0.44) ALDH1A1BCHETSHRL3MBTL1TDP1
SCHEMBL164228 0.72 BCHE (0.51) ALDH1A1BCHETSHRL3MBTL1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090325041-A1 Lithium Secondary Battery HITACHI, LTD. (JP) 2009-12-31 US disclosed
CN-1980660-A Contraceptive regimens and kits for progesterone receptor antagonists WYETH CORP (US) 2007-06-13 CN disclosed
EP-1351684-A4 COMPOUNDS AND METHODS FOR PROMOTING SMOKING CESSATION RES TRIANGLE INST (US) 2005-01-19 EP disclosed
WO-2005000806-A2 LIGANDS FOR NICOTINIC ACETYLCHOLINE RECEPTORS, AND METHODS OF MAKING AND USING THEM GEORGETOWN UNIVERSITY (US) 2005-01-06 WO disclosed
WO-2004099373-A2 BIOCOMPATIBLE RESISTS UNIVERSITY OF NORTH CAROLINA AT CHARLOTTE (US) 2004-11-18 WO disclosed
EP-1351684-A2 COMPOUNDS AND METHODS FOR PROMOTING SMOKING CESSATION Research Triangle Institute (US) 2003-10-15 EP disclosed
WO-2002037927-A2 COMPOUNDS AND METHODS FOR PROMOTING SMOKING CESSATION RESEARCH TRIANGLE INSTITUTE (US) 2002-05-16 WO disclosed
US-6384228-B2 EPIBATIDINE; ANALGESICS; ANIMAL EXTRACTS NIHON MEDI-PHYSICS CO., LTD. (JP) 2002-05-07 US disclosed
US-20020010339-A1 METHOD FOR SYNTHESIS OF HALOPYRIDYL-ACYCLOPENTANE DERIVATIVE AND INTERMEDIATE THEREOF NIHON MEDI-PHYSICS CO., LTD. (JP) 2002-01-24 US disclosed
US-5591854-A CATALYTIC CONDENSATION OF DIENES AND VINYLDIAZOMETHANEESTERS WAKE FOREST UNIVERSITY (US) 1997-01-07 US disclosed
WO-1996011928-A1 ENANTIOSELECTIVE SYNTHESIS OF SEVEN-MEMBERED CARBOCYCLES AND TROPANES WAKE FOREST UNIVERSITY (US) 1996-04-25 WO disclosed
US-3980089-A Novel heterocyclic flavoring compositions and processes INTERNATIONAL FLAVORS & FRAGRANCES INC. (US) 1976-09-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020010339-A1 METHOD FOR SYNTHESIS OF HALOPYRIDYL-ACYCLOPENTANE DERIVATIVE AND INTERMEDIATE THEREOF DHPS, ALAD, HAAO ALDH1A1 242/4885BCHE 2731/4885TSHR 4144/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.