SCHEMBL436808

SCHEMBL436808

CCCc1cc(N)c2cccc(C(F)(F)F)c2n1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSK P43235 4/20 0.45
CTSS P25774 3/20 0.44
MCHR1 Q99705 9/20 0.43
ACHE P22303 1/20 0.39
EIF4A1 P60842 1/20 0.39
KCNH2 Q12809 3/20 0.39
ESR1 P03372 1/20 0.39
PTPN1 P18031 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL436520 0.82 CYP2D6 (0.41) MCHR1KCNH2
SCHEMBL437914 0.81 CTSS (0.41) CTSKCTSSMCHR1
SCHEMBL439825 0.79 NR4A2 (0.60) MCHR1ACHE
SCHEMBL440380 0.79 ALDH1A1 (0.49) CTSKCTSSMCHR1EIF4A1
SCHEMBL30604783 0.77 KCNH2 (0.46) KCNH2ESR1
SCHEMBL30604781 0.77 KCNH2 (0.46) KCNH2ESR1
SCHEMBL438754 0.77 HSP90AB1 (0.52) MCHR1
SCHEMBL31690948 0.76 NR4A2 (0.47) ACHEKCNH2ESR1
SCHEMBL436015 0.74 NOS3 (0.39) CTSKCTSSMCHR1
SCHEMBL441586 0.72 KDM4E (0.60) MCHR1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed