SCHEMBL439825

SCHEMBL439825

CCCc1cc(N)c2cccc(Cl)c2n1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 3/20 0.60
HSP90AB1 P08238 1/20 0.50
MCHR1 Q99705 10/20 0.45
MAPT P10636 1/20 0.40
ACHE P22303 1/20 0.39
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
ASIC3 Q9UHC3 1/20 0.39
KDM4E B2RXH2 1/20 0.38
PARP1 P09874 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL436520 0.82 CYP2D6 (0.41) NR4A2MCHR1NOS3NOS1NOS2
SCHEMBL438225 0.82 MCHR1 (0.42) NR4A2MCHR1MAPTNOS3NOS1
SCHEMBL440380 0.82 ALDH1A1 (0.49) NR4A2MCHR1NOS3NOS1NOS2
SCHEMBL439885 0.81 NOS3 (0.41) NR4A2MCHR1NOS3NOS1NOS2
SCHEMBL439708 0.80 MCHR1 (0.43) NR4A2MCHR1MAPTACHENOS3
SCHEMBL436808 0.79 CTSK (0.45) MCHR1ACHE
SCHEMBL438754 0.79 HSP90AB1 (0.52) HSP90AB1MCHR1KDM4EPARP1
SCHEMBL438834 0.79 NOS2 (0.50) NR4A2HSP90AB1MCHR1MAPTNOS3
SCHEMBL436991 0.78 NOS3 (0.41) NR4A2HSP90AB1MCHR1MAPTNOS3
SCHEMBL438980 0.76 NR4A2 (1.00) NR4A2MAPTACHEKDM4EPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed