SCHEMBL437914

SCHEMBL437914

CCCc1cc(N)c2cccc(OC(F)(F)F)c2n1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.41
CTSK P43235 2/20 0.41
MPL P40238 1/20 0.40
MCHR1 Q99705 12/20 0.38
HSP90AB1 P08238 1/20 0.38
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
PDE10A Q9Y233 1/20 0.35
F2R P25116 1/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL438754 0.84 HSP90AB1 (0.52) MCHR1HSP90AB1PDE10A
SCHEMBL436808 0.81 CTSK (0.45) CTSSCTSKMCHR1
SCHEMBL437125 0.80 NR4A2 (0.55) MPLADORA2AADORA1
SCHEMBL436520 0.78 CYP2D6 (0.41) MCHR1ADORA2AADORA1NOS3NOS1
SCHEMBL440380 0.75 ALDH1A1 (0.49) CTSSCTSKMCHR1ADORA1NOS3
SCHEMBL439825 0.75 NR4A2 (0.60) MCHR1HSP90AB1NOS3NOS1NOS2
SCHEMBL441705 0.73 CTSS (0.45) CTSSCTSKMCHR1
SCHEMBL436437 0.73 MCHR1 (0.51) CTSSCTSKMCHR1
SCHEMBL436015 0.70 NOS3 (0.39) CTSSCTSKMCHR1NOS3NOS1
SCHEMBL441586 0.68 KDM4E (0.60) MCHR1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed