SCHEMBL438754

SCHEMBL438754

CCCc1cc(N)c2cccc(OC)c2n1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 1/20 0.52
KDM4E B2RXH2 4/20 0.44
MCHR1 Q99705 1/20 0.42
PDE10A Q9Y233 3/20 0.41
TLR8 Q9NR97 1/20 0.41
SREBF2 Q12772 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HSD17B10 Q99714 1/20 0.41
HTR1A P08908 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
TNKS O95271 1/20 0.40
PARP1 P09874 1/20 0.40
TNKS2 Q9H2K2 1/20 0.40
CYP3A4 P08684 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL437914 0.84 CTSS (0.41) HSP90AB1MCHR1PDE10A
SCHEMBL13409411 0.81 HSP90AB1 (0.44) HSP90AB1KDM4EPDE10ASREBF2ALDH1A1
SCHEMBL440380 0.79 ALDH1A1 (0.49) KDM4EMCHR1ALDH1A1HPGDTDP1
SCHEMBL436520 0.79 CYP2D6 (0.41) KDM4EMCHR1SMN1; SMN2TDP1
SCHEMBL439825 0.79 NR4A2 (0.60) HSP90AB1KDM4EMCHR1PARP1
SCHEMBL441787 0.79 MCHR1 (0.37) HSP90AB1MCHR1
SCHEMBL437287 0.77 NR4A2 (0.61) KDM4EMCHR1ALDH1A1HPGDSMN1; SMN2
SCHEMBL436808 0.77 CTSK (0.45) MCHR1
SCHEMBL18682211 0.74 PDE10A (0.68) MCHR1PDE10A
SCHEMBL23473307 0.72 KDM4E (0.51) HSP90AB1KDM4EPDE10AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed