SCHEMBL4373487

SCHEMBL4373487

NCCCC[C@H](C(N)=O)N(O)S(=O)(=O)c1ccc(Oc2ccc3c(c2)CCCC3)nc1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 15/20 0.44
OPRD1 P41143 15/20 0.44
OPRK1 P41145 12/20 0.44
HRH3 Q9Y5N1 3/20 0.42
MLNR O43193 1/20 0.39
CYP2D6 P10635 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4370947 0.88 OPRM1 (0.40) OPRM1OPRD1OPRK1HRH3MLNR
SCHEMBL1798242 0.77 MMP2 (0.42) OPRM1OPRD1OPRK1MLNRCYP2D6
SCHEMBL1800017 0.73 MMP2 (0.44) HTT
SCHEMBL1798723 0.67 ADAM17 (0.49)
SCHEMBL4375889 0.65 MAPK8 (0.35) ALDH1A1HTTNPSR1
SCHEMBL14878471 0.64 OPRM1 (0.41) OPRM1OPRD1OPRK1HRH3
SCHEMBL14380137 0.64 ALDH1A1 (0.57) OPRM1OPRD1OPRK1HRH3MLNR
SCHEMBL13604602 0.63 OPRM1 (0.46) OPRM1OPRD1OPRK1HRH3
SCHEMBL12653312 0.63 OPRM1 (0.46) OPRM1OPRD1OPRK1HRH3MLNR
SCHEMBL778932 0.62 NPC1 (0.49) OPRM1OPRD1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1461313-B1 HUMAN ADAM-10 INHIBITORS EXELIXIS INC (US) 2009-08-05 EP claimed
EP-1461313-B1 HUMAN ADAM-10 INHIBITORS EXELIXIS INC (US) 2009-08-05 EP disclosed