SCHEMBL439632

SCHEMBL439632

Cc1cc(N)c2ccc(OC(F)(F)F)cc2n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.54
NCF1 P14598 1/20 0.50
HSD17B10 Q99714 2/20 0.49
ALDH1A1 P00352 1/20 0.49
CASP1 P29466 1/20 0.49
CASP7 P55210 1/20 0.49
GNG2 P59768 2/20 0.46
GNB1 P62873 2/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
ALOX15 P16050 2/20 0.46
BLM P54132 2/20 0.46
GMNN O75496 1/20 0.46
USP2 O75604 1/20 0.46
LMNA P02545 1/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL439264 0.88 HSD17B10 (0.64) NR4A2NCF1HSD17B10ALDH1A1CASP1
SCHEMBL22828432 0.84 POLB (0.51) HSD17B10ALDH1A1NPC1RAB9AALOX15
SCHEMBL438970 0.81 NR4A2 (0.60) NR4A2NCF1HSD17B10ALDH1A1CASP1
SCHEMBL441705 0.79 CTSS (0.45) HSD17B10NPC1RAB9AALOX15BLM
SCHEMBL8180035 0.76 CYP1A2 (0.50) HSD17B10NPC1RAB9AALOX15BLM
SCHEMBL30682591 0.74 NR4A2 (0.64) NR4A2NCF1HSD17B10ALDH1A1CASP1
SCHEMBL442339 0.74 NR4A2 (0.64) NR4A2NCF1HSD17B10ALDH1A1CASP1
SCHEMBL28348548 0.73 GPR3 (0.51) HSD17B10NPC1RAB9AALOX15BLM
SCHEMBL21225586 0.72 PDE10A (0.46) HSD17B10NPC1RAB9AALOX15BLM
SCHEMBL32685110 0.71 CYP1A2 (0.52) NCF1HSD17B10NPC1RAB9AALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed