SCHEMBL439849

SCHEMBL439849

CCCc1cc(N)c2c(Cl)ccc(C)c2n1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.43
KDM4E B2RXH2 1/20 0.43
NOS2 P35228 3/20 0.41
NOS1 P29475 2/20 0.41
NOS3 P29474 1/20 0.41
MCHR1 Q99705 5/20 0.36
BACE1 P56817 1/20 0.36
CTSK P43235 3/20 0.35
MAPT P10636 3/20 0.34
TP53 P04637 1/20 0.34
LMNA P02545 2/20 0.34
HTT P42858 1/20 0.34
ASIC3 Q9UHC3 1/20 0.34
CTSS P25774 2/20 0.33
TLR7 Q9NYK1 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL436991 0.89 NOS3 (0.41) POLBNOS2NOS1NOS3MCHR1
SCHEMBL437233 0.78 NR4A2 (0.51) POLBKDM4EMAPTLMNAHTT
SCHEMBL439885 0.77 NOS3 (0.41) NOS2NOS1NOS3MCHR1BACE1
SCHEMBL441438 0.76 MAPT (0.43) KDM4ENOS2NOS1NOS3MCHR1
SCHEMBL438225 0.75 MCHR1 (0.42) POLBNOS2NOS1NOS3MCHR1
SCHEMBL439825 0.72 NR4A2 (0.60) KDM4ENOS2NOS1NOS3MCHR1
SCHEMBL438834 0.72 NOS2 (0.50) KDM4ENOS2NOS1NOS3MCHR1
SCHEMBL438887 0.72 MCHR1 (0.44) KDM4ENOS2NOS1NOS3MCHR1
SCHEMBL441901 0.70 MCHR1 (0.43) POLBKDM4ENOS2NOS1NOS3
SCHEMBL439708 0.70 MCHR1 (0.43) POLBNOS2NOS1NOS3MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed