SCHEMBL440033

SCHEMBL440033

Nc1c(C(=O)O)cnc2ccc(F)cc12

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.49
DHODH Q02127 3/20 0.47
ALDH1A1 P00352 3/20 0.46
GAA P10253 1/20 0.46
HAVCR2 Q8TDQ0 1/20 0.46
RXFP1 Q9HBX9 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
BCHE P06276 5/20 0.42
ACHE P22303 5/20 0.42
GRIN1 Q05586 5/20 0.42
GRIN2A Q12879 5/20 0.42
TP53 P04637 1/20 0.41
THRB P10828 1/20 0.41
PARP1 P09874 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL438745 0.88 KEAP1 (0.49) KEAP1DHODHALDH1A1GAAHAVCR2
SCHEMBL16621492 0.83 HAVCR2 (0.47) ALDH1A1HAVCR2KMT2AACHEPARP1
SCHEMBL398640 0.83 DHODH (0.47) KEAP1DHODHALDH1A1GAARXFP1
SCHEMBL22395713 0.81 DHODH (0.46) KEAP1DHODHALDH1A1GAARXFP1
SCHEMBL7496024 0.81 DHODH (0.46) KEAP1DHODHALDH1A1GAARXFP1
SCHEMBL440411 0.81 HAVCR2 (0.52) DHODHALDH1A1HAVCR2MEN1KMT2A
SCHEMBL442132 0.81 TSHR (0.50) DHODHALDH1A1GAAHAVCR2RXFP1
SCHEMBL436603 0.81 KDM4E (0.48) DHODHALDH1A1GAAHAVCR2MEN1
SCHEMBL439948 0.81 ALDH1A1 (0.53) DHODHALDH1A1HAVCR2MEN1KMT2A
SCHEMBL439008 0.79 NMT2 (0.60) ALDH1A1GAAMEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed