SCHEMBL4411527

SCHEMBL4411527

O=C(c1[c]cccc1)N1CCC(CO)C1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.45
VNN1 O95497 1/20 0.45
TACR3 P29371 1/20 0.44
AKR1C3 P42330 1/20 0.42
SPR P35270 2/20 0.40
HTR2C P28335 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
EPHX2 P34913 1/20 0.39
CYP2C9 P11712 3/20 0.39
CYP2C19 P33261 3/20 0.39
MAPK14 Q16539 3/20 0.39
HTR2B P41595 2/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4458413 0.81 PDK2 (0.43) PDK2VNN1NPC1RAB9A
SCHEMBL3984591 0.77 PDK1 (0.43) RAB9A
SCHEMBL4456609 0.77 L3MBTL3 (0.49) PDK2L3MBTL1
SCHEMBL1921739 0.77 L3MBTL1 (0.43) L3MBTL1SMN1; SMN2
SCHEMBL4352484 0.77 ACHE (0.59) NPC1RAB9ASMN1; SMN2
SCHEMBL28291394 0.77 CHRM2 (0.42) L3MBTL1CYP2C19RAB9ASMN1; SMN2
SCHEMBL4056659 0.74 PDK2 (0.38) PDK2VNN1NPC1RAB9A
SCHEMBL1115239 0.74 HPGD (0.47) NPC1SMN1; SMN2
SCHEMBL969710 0.74 HPGD (0.52) NPC1
SCHEMBL27804524 0.74 LMNA (0.56) NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664049-B1 SYNTHESIS OF PROTECTED PYRROLOBENZODIAZEPINES SPIROGEN LTD (GB) 2009-12-23 EP disclosed