SCHEMBL4412660

SCHEMBL4412660

Nc1[nH]c(Nc2ccc(Cc3ccncc3)cc2)nc2ncnc1-2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
CYP17A1 P05093 2/20 0.36
CYP19A1 P11511 2/20 0.36
CYP11B1 P15538 2/20 0.36
CYP11B2 P19099 2/20 0.36
CYP3A4 P08684 1/20 0.36
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.35
KMT2A Q03164 1/20 0.35
TDO2 P48775 1/20 0.35
HPGD P15428 3/20 0.35
MAPT P10636 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAPK1 P28482 3/20 0.34
LMNA P02545 2/20 0.34
METAP2 P50579 3/20 0.34
AURKB Q96GD4 1/20 0.34
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
LSS P48449 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4422876 0.81 PIK3CG (0.38) KMT2ANPC1RAB9AHTTSMN1; SMN2
SCHEMBL4414871 0.73 MAPT (0.45) ALDH1A1POLBKMT2AMAPTL3MBTL1
SCHEMBL350889 0.73 IRAK4 (0.41) ALDH1A1LMNAAURKBHTTSMN1; SMN2
SCHEMBL350890 0.73 IRAK4 (0.41) ALDH1A1LMNAAURKBHTTSMN1; SMN2
SCHEMBL4411964 0.71 TTBK1 (0.49) POLBMAPTMAPK1AURKBNPC1
SCHEMBL4428827 0.71 EGFR (0.50) MAPTNPC1RAB9AFLT1
SCHEMBL4417948 0.71 GAA (0.43) KMT2ATDO2MAPTL3MBTL1MAPK1
SCHEMBL4427810 0.70 EGFR (0.45) CYP3A4POLBTSHRKMT2AMAPT
SCHEMBL4414428 0.70 EGFR (0.47) TSHRMAPK1RAB9AHTTSMN1; SMN2
SCHEMBL4411564 0.70 CDC7 (0.49) ALDH1A1CYP3A4KMT2AHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7601713-B2 Kinase inhibitors and their uses RIGEL PHARMACEUTICALS, INC. (US) 2009-10-13 US claimed