SCHEMBL44400

SCHEMBL44400

O=S(=O)(NCc1cccc(-c2cn3ncccc3n2)c1)c1ccccc1Cl

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.41
SLC12A2 P55011 1/20 0.41
SLC12A5 Q9H2X9 1/20 0.41
PKM P14618 1/20 0.40
TP53 P04637 2/20 0.39
GLA P06280 1/20 0.39
CYP19A1 P11511 2/20 0.38
KMT2A Q03164 1/20 0.38
NR3C2 P08235 1/20 0.37
PIK3CD O00329 1/20 0.37
PIK3CG P48736 1/20 0.37
SLC40A1 Q9NP59 1/20 0.36
CNR1 P21554 1/20 0.36
POLB P06746 1/20 0.36
HSD11B1 P28845 1/20 0.36
WDR5 P61964 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL44570 0.88 CNR1 (0.40) LMNATP53CYP19A1KMT2ANR3C2
SCHEMBL44612 0.88 TSHR (0.42) ALDH1A1CYP19A1KMT2ANR3C2PIK3CD
SCHEMBL44344 0.84 TP53 (0.45) ALDH1A1LMNAPKMTP53CYP19A1
SCHEMBL44668 0.81 CYP19A1 (0.56) ALDH1A1LMNATP53CYP19A1KMT2A
SCHEMBL38873 0.78 CYP19A1 (0.47) ALDH1A1CYP19A1NR3C2PIK3CDPIK3CG
SCHEMBL12926166 0.78 PIK3CD (0.41) ALDH1A1TP53CYP19A1KMT2APIK3CD
SCHEMBL44258 0.77 CYP19A1 (0.60) ALDH1A1PKMCYP19A1KMT2APIK3CD
SCHEMBL22489884 0.76 PRMT6 (0.51) ALDH1A1LMNASLC12A2SLC12A5PKM
SCHEMBL44139 0.76 ALDH1A1 (0.43) ALDH1A1LMNASLC12A2SLC12A5TP53
SCHEMBL38716 0.74 FBP1 (0.47) ALDH1A1PIK3CDPIK3CGWDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO claimed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed