SCHEMBL4418740

SCHEMBL4418740

CNC(=O)OC(c1cn(S(=O)(=O)c2cccc(OC)c2)c(-c2cccnc2Cl)c1F)C(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.41
NFE2L2 Q16236 3/20 0.37
KAT8 Q9H7Z6 1/20 0.35
HTR6 P50406 6/20 0.34
ELAVL1 Q15717 1/20 0.33
GLO1 Q04760 1/20 0.33
SLC40A1 Q9NP59 1/20 0.33
ALPL P05186 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
FGFR4 P22455 2/20 0.32
ALDH1A1 P00352 1/20 0.32
PPARG P37231 1/20 0.32
PPARD Q03181 1/20 0.32
PPARA Q07869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2410874 0.92 NFE2L2 (0.35) METNFE2L2KAT8HTR6ALDH1A1
SCHEMBL4419026 0.89 MET (0.40) METNFE2L2KAT8HTR6ELAVL1
SCHEMBL2408730 0.88 NR3C1 (0.35) GLO1SLC40A1
SCHEMBL2408490 0.83 HTR6 (0.35) METHTR6FGFR4ALDH1A1DRD2
SCHEMBL4425656 0.83 MET (0.39) METALDH1A1
Hydrochloric Acid SCHEMBL4416301 0.82 MET (0.34) METHTR6ALPLFGFR4
SCHEMBL1834071 0.81 NFE2L2 (0.33) METNFE2L2ALDH1A1
SCHEMBL2410027 0.81 NTRK1 (0.31) ALDH1A1
SCHEMBL2409435 0.81 MET (0.43) METNFE2L2KAT8HTR6GLO1
SCHEMBL4425473 0.80 HTR6 (0.33) HTR6DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed