SCHEMBL4439796

SCHEMBL4439796

CC(C)(C)C(NC(=O)O)[C@H](Cc1ccccc1C(F)(F)F)NC(=O)c1ccc(Br)cn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
ANO1 Q5XXA6 2/20 0.37
TRPM8 Q7Z2W7 1/20 0.35
PPARG P37231 3/20 0.35
AKT1 P31749 1/20 0.35
AKT2 P31751 1/20 0.35
AKT3 Q9Y243 1/20 0.35
PPARA Q07869 1/20 0.35
EPHX2 P34913 2/20 0.35
SCN9A Q15858 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.35
GRM4 Q14833 1/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4431729 0.85 CCR1 (0.40) HDAC3HDAC1HDAC6KDM4EALDH1A1
SCHEMBL4553919 0.82 AKT1 (0.38) ANO1AKT1SCN9ASCN10AMEN1
SCHEMBL4380618 0.81 ALDH1A1 (0.41) ANO1PPARGAKT1AKT2AKT3
SCHEMBL4382045 0.79 EPHX2 (0.37) ANO1PPARGAKT1AKT2AKT3
SCHEMBL4379890 0.79 AKT1 (0.43) PPARGAKT1AKT2AKT3PPARA
SCHEMBL4376050 0.78 AKT1 (0.44) HDAC3HDAC1HDAC2HDAC6ANO1
SCHEMBL3333499 0.78 HDAC3 (0.39) HDAC3HDAC1HDAC2HDAC6ANO1
SCHEMBL3333495 0.78 HDAC3 (0.39) HDAC3HDAC1HDAC2HDAC6ANO1
SCHEMBL13300019 0.75 SCN9A (0.42) HDAC3HDAC1HDAC2HDAC6AKT1
SCHEMBL4543991 0.74 AKT1 (0.45) AKT1AKT2AKT3EPHX2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2134175-A1 INHIBITORS OF AKT ACTIVITY Smithkline Beecham Corporation (US) 2009-12-23 EP disclosed
WO-2008121786-A1 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2008-10-09 WO disclosed