SCHEMBL4453396

SCHEMBL4453396

Nc1nc2c(Cc3cccc4c3OCCO4)cc(-c3ccncc3F)cc2s1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
ROCK2 O75116 2/20 0.34
ROCK1 Q13464 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
LMNA P02545 3/20 0.32
TP53 P04637 2/20 0.32
PIK3CD O00329 1/20 0.31
PIP5K1C O60331 1/20 0.31
PIK3CA P42336 1/20 0.31
PI4KA P42356 1/20 0.31
PI4KB Q9UBF8 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4285908 0.73 ROCK2 (0.44) ROCK2ROCK1CYP3A4CYP2D6CYP2C9
SCHEMBL20855280 0.62 ABL1 (0.57) SMN1; SMN2LMNAPIK3CDPIP5K1CPIK3CA
SCHEMBL4284870 0.59 ROCK2 (0.60) ROCK2ROCK1CYP3A4CYP2D6CYP2C9
SCHEMBL4555423 0.58 MPO (0.44) ROCK2ROCK1SMN1; SMN2LMNAALDH1A1
SCHEMBL8548188 0.58 RAB9A (0.51) CYP3A4LMNAPIK3CDPIP5K1CPIK3CA
SCHEMBL29078645 0.58 HSD17B10 (0.53) CYP3A4CYP2D6CYP2C9PIK3CDPIP5K1C
SCHEMBL1010573 0.57 MTNR1A (0.55) ADORA2AADORA1ROCK2ROCK1CYP3A4
SCHEMBL2944410 0.56 ALDH1A1 (0.45) ADORA2AADORA1CYP3A4CYP2D6SMN1; SMN2
SCHEMBL3749352 0.56 ADRA1D (0.51) CYP3A4CYP2D6SMN1; SMN2
SCHEMBL31407536 0.56 MTNR1A (0.53) ADORA2AADORA1ROCK2ROCK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009126635-A1 2-AMINO-BENZOTHIAZOLE DERIVATES USEFUL AS INHIBITORS OF ROCK KINASES ABBOTT LABORATORIES (US) 2009-10-15 WO disclosed