SCHEMBL446622

SCHEMBL446622

Cc1cc(C)c(B(O)O)c(-c2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.47
PSMB5 P28074 3/20 0.42
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MCOLN3 Q8TDD5 1/20 0.40
METAP2 P50579 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
BACE1 P56817 1/20 0.39
ALOX5 P09917 1/20 0.38
NUDT1 P36639 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37
MGLL Q99685 2/20 0.37
CYP2A6 P11509 2/20 0.37
CYP2B6 P20813 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
ALDH1A1 P00352 2/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4438197 0.92 ESR2 (0.41) ESR2PSMB5LMNASMN1; SMN2MCOLN3
SCHEMBL448143 0.79 CA2 (0.43) LMNACYP2A6CA1CA2ALDH1A1
SCHEMBL431299 0.78 MGLL (0.48) ESR2SMN1; SMN2ALOX5MGLLCA1
SCHEMBL30255125 0.77 PDCD1 (0.44) ESR2SMN1; SMN2BACE1MGLLCYP2A6
SCHEMBL8986922 0.75 ESR2 (0.52) ESR2PSMB5LMNASMN1; SMN2MCOLN3
SCHEMBL24665564 0.74 MGLL (0.48) ESR2LMNASMN1; SMN2BACE1ALOX5
SCHEMBL9423370 0.74 PSMB5 (0.49) ESR2PSMB5LMNASMN1; SMN2MCOLN3
SCHEMBL19464511 0.73 HDAC7 (0.49) ESR2PSMB5LMNAMETAP2HDAC7
Water SCHEMBL19349803 0.72 PSMB5 (0.47) ESR2PSMB5LMNASMN1; SMN2MCOLN3
SCHEMBL2528210 0.71 BACE1 (0.54) ESR2PSMB5METAP2HDAC7BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115490607-A C 2 Synthesis method of-symmetrical chiral aryl iodide catalyst 南通大学 2022-12-20 CN disclosed
US-8536351-B2 2-aryl-5-heterocyclyl-cyclohexane-1,3,dione compounds and their use as herbicides SYNGENTA CROP PROTECTION LLC (US) 2013-09-17 US disclosed
EP-2429979-A1 NOVEL HERBICIDES Syngenta Limited (GB) 2012-03-21 EP disclosed
US-20120065066-A1 NOVEL HERBICIDES SYNGENTA CROP PROTECTION LLC (US) 2012-03-15 US disclosed
US-8084649-B2 Herbicides SYNGENTA CROP PROTECTION, INC. (US) 2011-12-27 US disclosed
EP-2134699-B1 2-ARYL-5-HETEROCYCLYL-CYCLOHEXANE-1,3-DIONE COMPOUNDS AND THEIR USE AS HERBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2011-05-11 EP disclosed
WO-2010133232-A1 NOVEL HERBICIDES SYNGENTA LIMITED (GB) 2010-11-25 WO disclosed
US-20100173774-A1 NOVEL HERBICIDES SYNGENTA CROP PROTECTION, INC. (US) 2010-07-08 US disclosed
US-20100113270-A1 2-ARYL-5-HETEROCYCLYL-CYCLOHEXANE-1,3,DIONE COMPOUNDS AND THEIR USE AS HERBICIDES SYNGENTA CROP PROTECTION, INC. (US) 2010-05-06 US disclosed
EP-2134699-A1 2-ARYL-5-HETEROCYCLYL-CYCLOHEXANE-1,3-DIONE COMPOUNDS AND THEIR USE AS HERBICIDES Syngeta Participations AG (CH) 2009-12-23 EP disclosed
EP-2121584-A2 NOVEL HERBICIDES Syngeta Participations AG (CH) 2009-11-25 EP disclosed
WO-2008110307-A1 2-ARYL-5-HETEROCYCLYL-CYCLOHEXANE-1,3-DIONE COMPOUNDS AND THEIR USE AS HERBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2008-09-18 WO disclosed
WO-2008110308-A2 NOVEL HERBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2008-09-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120065066-A1 NOVEL HERBICIDES DDT, CYP4X1, CYP1B1 ESR2 1787/4885PSMB5 2872/4885LMNA 4657/4885
US-20100113270-A1 2-ARYL-5-HETEROCYCLYL-CYCLOHEXANE-1,3,DIONE COMPOUNDS AND THEIR USE AS HERBICIDES C3AR1, C5, C9 ESR2 517/4885PSMB5 1083/4885LMNA 1709/4885
US-20100173774-A1 NOVEL HERBICIDES DDT, HDHD5, HPD ESR2 1428/4885PSMB5 1811/4885LMNA 4588/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.