SCHEMBL44668

SCHEMBL44668

O=S(=O)(NCc1cccc(-c2cn3ncccc3n2)c1)c1ccc(F)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 9/20 0.56
CNR1 P21554 1/20 0.45
LMNA P02545 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
TP53 P04637 2/20 0.41
POLB P06746 2/20 0.41
KIT P10721 1/20 0.41
NAMPT P43490 1/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL44570 0.85 CNR1 (0.40) CYP19A1CNR1LMNAKMT2ATP53
SCHEMBL44344 0.85 TP53 (0.45) CYP19A1LMNAALDH1A1MEN1KMT2A
SCHEMBL44258 0.84 CYP19A1 (0.60) CYP19A1ALDH1A1MEN1KMT2ACA1
SCHEMBL38873 0.82 CYP19A1 (0.47) CYP19A1ALDH1A1NAMPTPIK3CDPIK3CG
SCHEMBL12926166 0.82 PIK3CD (0.41) CYP19A1ALDH1A1MEN1KMT2ATP53
SCHEMBL44417 0.81 CYP19A1 (0.39) CYP19A1LMNAMEN1KMT2ATP53
SCHEMBL44612 0.81 TSHR (0.42) CYP19A1KDM4EALDH1A1HPGDMEN1
SCHEMBL44400 0.81 ALDH1A1 (0.45) CYP19A1CNR1LMNAALDH1A1KMT2A
SCHEMBL38716 0.77 FBP1 (0.47) KDM4EALDH1A1NAMPTMAPTPIK3CD
SCHEMBL39342 0.75 CYP19A1 (0.53) CYP19A1CNR1LMNAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO claimed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed