SCHEMBL44344

SCHEMBL44344

O=S(=O)(NCc1cccc(-c2cn3ncccc3n2)c1)c1cccc(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.45
CYP19A1 P11511 3/20 0.44
PIK3CD O00329 1/20 0.42
PIK3CG P48736 1/20 0.42
HSD11B1 P28845 7/20 0.42
ALDH1A1 P00352 1/20 0.42
PKM P14618 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
KDM1A O60341 1/20 0.41
MAOA P21397 1/20 0.41
LMNA P02545 1/20 0.41
AKT1 P31749 1/20 0.41
NAMPT P43490 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38873 0.85 CYP19A1 (0.47) CYP19A1PIK3CDPIK3CGALDH1A1NAMPT
SCHEMBL12926166 0.85 PIK3CD (0.41) TP53CYP19A1PIK3CDPIK3CGALDH1A1
SCHEMBL44668 0.85 CYP19A1 (0.56) TP53CYP19A1PIK3CDPIK3CGALDH1A1
SCHEMBL44258 0.85 CYP19A1 (0.60) CYP19A1PIK3CDPIK3CGALDH1A1PKM
SCHEMBL44400 0.84 ALDH1A1 (0.45) TP53CYP19A1PIK3CDPIK3CGHSD11B1
SCHEMBL44519 0.83 LMNA (0.42) TP53HSD11B1ALDH1A1PKMSMN1; SMN2
SCHEMBL44570 0.80 CNR1 (0.40) TP53CYP19A1PIK3CDPIK3CGLMNA
SCHEMBL44612 0.80 TSHR (0.42) CYP19A1PIK3CDPIK3CGALDH1A1SMN1; SMN2
SCHEMBL38716 0.77 FBP1 (0.47) PIK3CDPIK3CGALDH1A1SMN1; SMN2NAMPT
SCHEMBL22489791 0.76 NAMPT (0.54) TP53CYP19A1HSD11B1ALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO claimed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed