SCHEMBL4486859

SCHEMBL4486859

Cc1cc(C(N)=O)ccc1-c1ccc(CNCc2cccc(F)c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.52
OPRD1 P41143 2/20 0.52
OPRK1 P41145 2/20 0.52
MAOB P27338 3/20 0.44
PARP10 Q53GL7 1/20 0.44
KLKB1 P03952 1/20 0.43
PARP1 P09874 1/20 0.43
SRC P12931 1/20 0.43
CDC7 O00311 1/20 0.43
ROCK2 O75116 1/20 0.43
MAP4K4 O95819 1/20 0.43
PIM1 P11309 1/20 0.43
CDK2 P24941 1/20 0.43
GSK3B P49841 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
GPR52 Q9Y2T5 2/20 0.42
PPARA Q07869 1/20 0.41
CHEK2 O96017 1/20 0.41
SCN8A Q9UQD0 1/20 0.40
MAOA P21397 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4487434 0.88 SMN1; SMN2 (0.50) OPRM1OPRD1OPRK1PPARA
SCHEMBL4074391 0.86 HDAC1 (0.56) PARP1ROCK2GPR52
SCHEMBL4073993 0.83 SCN3A (0.42) MAOBPARP10CHEK2
SCHEMBL1788221 0.82 OPRM1 (0.54) OPRM1OPRD1OPRK1MAOBPARP10
SCHEMBL4074968 0.81 OPRM1 (0.60) OPRM1OPRD1OPRK1
SCHEMBL4081861 0.79 OPRM1 (0.53) OPRM1OPRD1OPRK1
SCHEMBL4073644 0.77 OPRM1 (0.53) OPRM1OPRD1OPRK1
Trifluoroacetic Acid SCHEMBL3340260 0.76 SRC (0.50) OPRM1OPRD1OPRK1PARP1SRC
Hydrochloric Acid SCHEMBL4073979 0.76 OPRM1 (0.52) OPRM1OPRD1OPRK1
SCHEMBL4075498 0.76 OPRM1 (0.43) OPRM1OPRD1OPRK1ROCK2MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7615651-B2 Diaryl, dipyridinyl and aryl-pyridinyl derivatives and uses thereof PFIZER INC. (US) 2009-11-10 US claimed