SCHEMBL4487434

SCHEMBL4487434

Cc1cc(C(N)=O)ccc1-c1ccc(CNCc2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.50
HDAC8 Q9BY41 2/20 0.48
HDAC6 Q9UBN7 1/20 0.48
OPRM1 P35372 2/20 0.47
OPRD1 P41143 2/20 0.47
OPRK1 P41145 2/20 0.47
RARB P10826 1/20 0.47
PLA2G10 O15496 1/20 0.45
PLA2G2A P14555 1/20 0.45
EGFR P00533 1/20 0.45
HDAC1 Q13547 1/20 0.44
AR P10275 1/20 0.43
ADRB1 P08588 1/20 0.43
ADRB3 P13945 1/20 0.43
DGAT1 O75907 2/20 0.42
SOAT1 P35610 2/20 0.42
MAPK14 Q16539 1/20 0.42
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4074968 0.92 OPRM1 (0.60) OPRM1OPRD1OPRK1RARBHDAC1
SCHEMBL4081861 0.90 OPRM1 (0.53) SMN1; SMN2HDAC8HDAC6OPRM1OPRD1
SCHEMBL4074391 0.88 HDAC1 (0.56) HDAC1ADRB1ADRB3PPARGALDH1A1
SCHEMBL4486859 0.88 OPRM1 (0.52) OPRM1OPRD1OPRK1PPARA
SCHEMBL4073993 0.87 SCN3A (0.42) SMN1; SMN2RARBHDAC1ALDH1A1HPGD
SCHEMBL4498120 0.85 HDAC1 (0.53) SMN1; SMN2HDAC8HDAC6OPRM1OPRD1
SCHEMBL4075498 0.84 OPRM1 (0.43) HDAC6OPRM1OPRD1OPRK1RARB
SCHEMBL2026285 0.83 ESR2 (0.55) RARBPPARGPPARAALDH1A1HPGD
SCHEMBL4073644 0.83 OPRM1 (0.53) SMN1; SMN2OPRM1OPRD1OPRK1RARB
Hydrochloric Acid SCHEMBL4073979 0.82 OPRM1 (0.52) SMN1; SMN2OPRM1OPRD1OPRK1RARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7615651-B2 Diaryl, dipyridinyl and aryl-pyridinyl derivatives and uses thereof PFIZER INC. (US) 2009-11-10 US claimed