SCHEMBL4487479

SCHEMBL4487479

CCc1c(C(=O)O)c(C=O)n(C)c1-c1nccs1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
ESR1 P03372 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HSF1 Q00613 1/20 0.31
GRIK1 P39086 1/20 0.31
GRIA1 P42261 1/20 0.31
GRIA2 P42262 1/20 0.31
GRIA3 P42263 1/20 0.31
GRIA4 P48058 1/20 0.31
GRIK2 Q13002 1/20 0.31
GRIK3 Q13003 1/20 0.31
GRIK4 Q16099 1/20 0.31
GRIK5 Q16478 1/20 0.31
ADORA3 P0DMS8 2/20 0.30
ADORA2A P29274 2/20 0.30
ADORA1 P30542 2/20 0.30
ADORA2B P29275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4492339 0.78 MAPT (0.34) SMN1; SMN2
SCHEMBL4488653 0.76 ERCC1 (0.38)
SCHEMBL4498679 0.75 CCNC (0.36) SMN1; SMN2HDAC3HDAC1HDAC6
SCHEMBL4504195 0.74 CCR1 (0.38) SMN1; SMN2
SCHEMBL4491009 0.73 ALDH1A1 (0.43) SMN1; SMN2GRIA2GRIA4
SCHEMBL4491753 0.73 POLB (0.35) SMN1; SMN2ADORA3ADORA2AADORA1
SCHEMBL4490745 0.70 GRIA2 (0.40) GRIA2GRIA4
SCHEMBL4480912 0.69
SCHEMBL4496740 0.69 GRM5 (0.39) ADORA3
SCHEMBL4488870 0.68 MEN1 (0.43) SMN1; SMN2GRIA2GRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504429-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2009-03-17 US claimed