SCHEMBL4488653

SCHEMBL4488653

CCc1c(C(=O)O)c(C=O)n(C)c1-c1cccs1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 1/20 0.38
FEN1 P39748 1/20 0.38
ERCC4 Q92889 1/20 0.38
ALDH1A1 P00352 9/20 0.37
KDM4E B2RXH2 9/20 0.37
MEN1 O00255 6/20 0.37
KMT2A Q03164 6/20 0.37
POLB P06746 5/20 0.37
HSD17B10 Q99714 3/20 0.37
HPGD P15428 3/20 0.37
ALOX15 P16050 2/20 0.37
TSHR P16473 2/20 0.37
CASP1 P29466 2/20 0.37
CASP7 P55210 2/20 0.37
USP2 O75604 2/20 0.37
GAA P10253 2/20 0.37
GFER P55789 1/20 0.37
PKM P14618 1/20 0.36
DPP4 P27487 1/20 0.35
NPC1 O15118 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4491009 0.80 ALDH1A1 (0.43) ALDH1A1KDM4EPOLBHSD17B10HPGD
SCHEMBL4492339 0.79 MAPT (0.34) ALDH1A1KDM4EMEN1KMT2APOLB
SCHEMBL4498679 0.76 CCNC (0.36) ALDH1A1KDM4EPOLBHPGDRAB9A
SCHEMBL4487479 0.76 ECE1 (0.33)
SCHEMBL4490745 0.74 GRIA2 (0.40) ALDH1A1KDM4EKMT2AHSD17B10ALOX15
SCHEMBL4492957 0.72 GRIA2 (0.42) ALDH1A1KDM4EMEN1KMT2AHSD17B10
SCHEMBL4496740 0.72 GRM5 (0.39) KDM4EMEN1KMT2APOLBNPC1
SCHEMBL4488870 0.72 MEN1 (0.43) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL4489152 0.72 TDP1 (0.44) NPC1RAB9ATDP1L3MBTL1
SCHEMBL4491753 0.72 POLB (0.35) KDM4EMEN1KMT2APOLBNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504429-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2009-03-17 US claimed