SCHEMBL4515089

SCHEMBL4515089

Cc1cccc(-c2ccccc2Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.58
MAPK14 Q16539 1/20 0.45
TNKS2 Q9H2K2 1/20 0.45
CLK4 Q9HAZ1 2/20 0.45
HSD11B1 P28845 2/20 0.44
ACHE P22303 1/20 0.44
SCN9A Q15858 1/20 0.43
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43
PLA2G7 Q13093 1/20 0.43
ENPP3 O14638 1/20 0.43
NPC1 O15118 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CNR2 P34972 2/20 0.42
CNR1 P21554 1/20 0.42
AKR1C2 P52895 1/20 0.42
AKR1C1 Q04828 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8817721 0.86 ACHE (0.42) CYP2A6MAPK14CLK4ACHESCN9A
SCHEMBL9479255 0.84 CYP2A6 (0.71) CYP2A6TNKS2HSD11B1SCN9ANPC1
SCHEMBL29628996 0.84 CYP2A6 (0.71) CYP2A6TNKS2HSD11B1SCN9ANPC1
SCHEMBL28414965 0.84 ACHE (0.55) CLK4ACHEKMT2AENPP3NPC1
SCHEMBL24689747 0.82 ACHE (0.52) CLK4ACHEKMT2AENPP3NPC1
SCHEMBL2922149 0.80 RAB9A (0.52) CLK4ACHEKMT2AENPP3NPC1
SCHEMBL10703217 0.80 DPP4 (0.52) HSD11B1NPC1HPGDTSHRRAB9A
SCHEMBL12431877 0.79 BACE1 (0.53) CYP2A6TNKS2HSD11B1KMT2AABL1
SCHEMBL5025375 0.78 HTR7 (0.55) CLK4ACHEPOLBKMT2AENPP3
SCHEMBL23759509 0.78 CYP2A6 (0.70) CYP2A6HSD11B1SCN9ANPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118852231-A Heterogeneous palladium-catalyzed C (sp2) -H bond silylation reaction 哈尔滨工业大学(深圳)(哈尔滨工业大学深圳科技创新研究院) 2024-10-29 CN disclosed
CN-107987034-A Preparation method of dibenzo [ c, e ] [1,2] thiazine-5-oxo series compound with tricyclic system structure 江西师范大学 2018-05-04 CN disclosed
EP-2570418-A2 2,3-dihydro-6-nitroimidazo[2,1-b]oxazoles compound OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2013-03-20 EP disclosed
EP-1555267-B1 2,3-DIHYDRO-6-NITROIMIDAZO[2,1-b]OXAZOLES OTSUKA PHARMA CO LTD (JP) 2013-01-16 EP disclosed
US-20120135997-A1 PHARMACEUTICAL COMPOSITION COMPRISING A LACTAM OR BENZENESULFONAMIDE COMPOUND SHIONOGI & CO., LTD. (JP) 2012-05-31 US disclosed
US-8044068-B2 Aminopyrrolidine compound TAISHO PHARMACEUTICAL CO., LTD (JP) 2011-10-25 US disclosed
US-8044068-B2 Aminopyrrolidine compound TAISHO PHARMACEUTICAL CO., LTD (JP) 2011-10-25 US disclosed
WO-2011007819-A1 PHARMACEUTICAL PRODUCT CONTAINING LACTAM OR BENZENE SULFONAMIDE COMPOUND 塩野義製薬株式会社 (JP) 2011-01-20 WO disclosed
US-20090291940-A1 AMINOPYRROLIDINE COMPOUND TAISHO PHARMACEUTICAL CO., LTD. (JP) 2009-11-26 US disclosed
US-20090291940-A1 AMINOPYRROLIDINE COMPOUND TAISHO PHARMACEUTICAL CO., LTD. (JP) 2009-11-26 US disclosed
US-20090275581-A1 RENIN INHIBITORS VITAE PHARMACEUTICALS, INC. 2009-11-05 US disclosed
EP-2003131-A1 AMINOPYRROLIDINE COMPOUND Taisho Pharmaceutical Co. Ltd. (JP) 2008-12-17 EP disclosed
WO-2008001160-A1 MELANIN CONCENTRATING HORMONE ANTAGONISTS THE PROCTER & GAMBLE COMPANY (US) 2008-01-03 WO disclosed
EP-1847533-A1 SIX-MEMBERED HETEROCYCLIC COMPOUND AND THE USE THEREOF Asahi Kasei Pharma Corporation (JP) 2007-10-24 EP disclosed
US-7262212-B2 2,3-dihydro-6-nitroimidazo[2,1-b]oxazoles OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-08-28 US disclosed
US-20060094767-A1 2,3-Dihydro-6-nitroimidazo[2,1-b]oxazoles OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-05-04 US disclosed
EP-1555267-A1 2,3-DIHYDRO-6-NITROIMIDAZO 2,1-b OXAZOLES OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2005-07-20 EP disclosed
EP-0342532-A1 Process for the preparation of 4-chloro-2-methyl-5-nitro-phenol Wella Aktiengesellschaft (DE) 1989-11-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120135997-A1 PHARMACEUTICAL COMPOSITION COMPRISING A LACTAM OR BENZENESULFONAMIDE COMPOUND BACE1, STS, APP CYP2A6 470/4885MAPK14 4702/4885TNKS2 4467/4885
US-20060094767-A1 2,3-Dihydro-6-nitroimidazo[2,1-b]oxazoles NR2C2, NR4A3, NR4A2 CYP2A6 1119/4885MAPK14 2803/4885TNKS2 3109/4885
US-20090275581-A1 RENIN INHIBITORS REN, ACE, SERPINB1 CYP2A6 1824/4885MAPK14 1632/4885TNKS2 4552/4885
US-20090291940-A1 AMINOPYRROLIDINE COMPOUND MC4R, MC5R, MC2R CYP2A6 3620/4885MAPK14 616/4885TNKS2 3320/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.