SCHEMBL4523904

SCHEMBL4523904

CC(C)Oc1ccc(COc2ccc(CCCO)cc2)cc1

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.67
EPHX2 P34913 1/20 0.67
SIGMAR1 Q99720 1/20 0.50
BCHE P06276 2/20 0.46
KDM4E B2RXH2 1/20 0.46
POLB P06746 1/20 0.45
ACACB O00763 2/20 0.44
FFAR1 O14842 2/20 0.43
PPARA Q07869 1/20 0.43
LMNA P02545 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
RXRA P19793 1/20 0.42
RXRB P28702 1/20 0.42
FFAR4 Q5NUL3 1/20 0.42
MCL1 Q07820 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5355098 0.90 POLB (0.53) LTA4HEPHX2KDM4EPOLBACACB
SCHEMBL11683841 0.89 POLB (0.51) LTA4HEPHX2KDM4EPOLBACACB
SCHEMBL23266258 0.85 POLB (0.51) LTA4HEPHX2KDM4EPOLBACACB
SCHEMBL4508064 0.84 SIGMAR1 (0.47) LTA4HEPHX2SIGMAR1BCHEKDM4E
SCHEMBL9112221 0.83 POLB (0.50) LTA4HEPHX2KDM4EPOLBACACB
SCHEMBL9027085 0.83 POLB (0.50) LTA4HEPHX2KDM4EPOLBACACB
SCHEMBL5174164 0.82 BCHE (0.47) BCHEKDM4EPOLBLMNAL3MBTL1
SCHEMBL14033258 0.82 LTA4H (0.73) LTA4HEPHX2SIGMAR1FFAR1PPARA
SCHEMBL29886710 0.82 LTA4H (0.73) LTA4HEPHX2BCHEPOLBFFAR1
SCHEMBL3172997 0.82 APP (0.59) BCHEPOLBPPARALMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1527065-B1 METHOD FOR THE PRODUCTION OF (S)-3-METHYLAMINO-1-(THIEN-2-YL)PROPAN-1-OL BASF AG (DE) 2006-11-22 EP claimed
US-7498460-B2 Isophthalic acid derivatives BAYER HEALTHCARE AG (DE) 2009-03-03 US disclosed
US-7498460-B2 Isophthalic acid derivatives BAYER HEALTHCARE AG (DE) 2009-03-03 US disclosed
US-7498460-B2 Isophthalic acid derivatives BAYER HEALTHCARE AG (DE) 2009-03-03 US disclosed
US-7435563-B2 Method for the production of (s)-3-methylamino-1-(thien-2-yl)propan-1-ol BASF AKTIENGESELLSCHAFT (DE) 2008-10-14 US disclosed
US-20080176898-A1 Leukotriene antagonists; cardiovascular disorders like unstable angina pectoris or myocardial infarction; Methyl 1-{[5-(ethoxycarbonyl)-2-(3-{4-[(4-isopropoxybenzyl)oxy]phenyl}propoxy)phenyl]-acetyl}piperidine-4-carboxylate BAYER HEALTHCARE AG (DE) 2008-07-24 US disclosed
US-20080176898-A1 Leukotriene antagonists; cardiovascular disorders like unstable angina pectoris or myocardial infarction; Methyl 1-{[5-(ethoxycarbonyl)-2-(3-{4-[(4-isopropoxybenzyl)oxy]phenyl}propoxy)phenyl]-acetyl}piperidine-4-carboxylate BAYER HEALTHCARE AG (DE) 2008-07-24 US disclosed
US-20080176898-A1 Leukotriene antagonists; cardiovascular disorders like unstable angina pectoris or myocardial infarction; Methyl 1-{[5-(ethoxycarbonyl)-2-(3-{4-[(4-isopropoxybenzyl)oxy]phenyl}propoxy)phenyl]-acetyl}piperidine-4-carboxylate BAYER HEALTHCARE AG (DE) 2008-07-24 US disclosed
EP-1572628-B1 ISOPHTALIC ACID DERIVATIVES BAYER HEALTHCARE AG (DE) 2007-07-25 EP disclosed
EP-1572628-B1 ISOPHTALIC ACID DERIVATIVES BAYER HEALTHCARE AG (DE) 2007-07-25 EP disclosed
EP-1740540-A1 PHENYL ACETAMIDES Bayer HealthCare AG (DE) 2007-01-10 EP disclosed
US-20060154912-A1 Isophtalic acid derivatives BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2006-07-13 US disclosed
WO-2005103001-A1 PHENYL ACETAMIDES BAYER HEALTHCARE AG (DE) 2005-11-03 WO disclosed
US-20050245749-A1 Method for the production of (s)-3-methylamino-1-(thien-2-yl)propan-1-ol BASF AKTIENGESELLSCHAFT (DE) 2005-11-03 US disclosed
EP-1572628-A1 ISOPHTALIC ACID DERIVATIVES Bayer HealthCare AG (DE) 2005-09-14 EP disclosed
WO-2004052839-A1 ISOPHTALIC ACID DERIVATIVES BAYER HEALTHCARE AG (DE) 2004-06-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080176898-A1 Leukotriene antagonists; cardiovascular disorders like unstable angina pectoris or myocardial infarction; Methyl 1-{[5-(ethoxycarbonyl)-2-(3-{4-[(4-isopropoxybenzyl)oxy]phenyl}propoxy)phenyl]-acetyl}piperidine-4-carboxylate LTC4S, LTB4R2, LTB4R LTA4H 6/4885EPHX2 1210/4885SIGMAR1 2420/4885
US-20050245749-A1 Method for the production of (s)-3-methylamino-1-(thien-2-yl)propan-1-ol INMT, PNMT, TH LTA4H 2271/4885EPHX2 692/4885SIGMAR1 572/4885
US-20060154912-A1 Isophtalic acid derivatives VHL, FABP3, CPT1A LTA4H 281/4885EPHX2 214/4885SIGMAR1 4200/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.