SCHEMBL453605

SCHEMBL453605

COc1c(F)ccc(C=O)c1OC

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
ALDH1A1 P00352 3/20 0.41
ERN1 O75460 10/20 0.40
TRIM24 O15164 1/20 0.40
TYR P14679 1/20 0.40
TRIM33 Q9UPN9 1/20 0.40
MCL1 Q07820 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
KDM4E B2RXH2 1/20 0.38
TSHR P16473 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
SRC P12931 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29729025 0.87 CA1 (0.59) CA1CA2ALDH1A1ERN1TRIM24
SCHEMBL3345839 0.87 CA1 (0.59) CA1CA2ALDH1A1ERN1TRIM24
SCHEMBL31538163 0.86 CA1 (0.47) CA1CA2ALDH1A1ERN1TRIM24
SCHEMBL1238926 0.86 CA1 (0.43) CA1CA2ALDH1A1ERN1TRIM24
SCHEMBL3256940 0.82 CA1 (0.41) CA1CA2ALDH1A1ERN1TRIM24
SCHEMBL16411961 0.82 CA1 (0.41) CA1CA2ALDH1A1ERN1TRIM24
SCHEMBL16187926 0.82 ERN1 (0.53) CA1CA2ERN1TRIM24TYR
SCHEMBL9894251 0.82 ERN1 (0.53) CA1CA2ERN1TRIM24TYR
SCHEMBL680844 0.82 CA1 (0.61) CA1CA2ALDH1A1ERN1MCL1
SCHEMBL9873091 0.79 KDM4E (0.43) CA1CA2ALDH1A1KDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220184236-A1 NANOPARTICLE, CONTRAST AGENT FOR MAGNETIC RESONANCE IMAGING COMPRISING SAME AND ZWITTERIONIC LIGAND COMPOUND National Institutes for Quantum Science and Technology (JP) 2022-06-16 US disclosed
US-20220089455-A1 METHOD FOR PRODUCING NANOPARTICLE HAVING METAL PARTICLE WHICH CONTAINS IRON OXIDE TO WHICH ONE OR MORE HYDROPHILIC LIGANDS ARE COORDINATION BONDED ASTELLAS PHARMA INC. (JP) 2022-03-24 US disclosed
EP-3904294-A1 METHOD FOR PRODUCING NANOPARTICLES INCLUDING METAL PARTICLES CONTAINING IRON OXIDE HAVING AT LEAST ONE HYDROPHILIC LIGAND COORDINATED THERETO Astellas Pharma Inc. (JP) 2021-11-03 EP disclosed
EP-3904331-A1 NANOPARTICLE, CONTRAST AGENT FOR MAGNETIC RESONANCE IMAGING COMPRISING SAME AND ZWITTERIONIC LIGAND COMPOUND Astellas Pharma Inc. (JP) 2021-11-03 EP disclosed
CN-113227040-A Nanoparticles, nuclear magnetic resonance imaging contrast agent containing nanoparticles and zwitterionic ligand compound 安斯泰来制药株式会社 2021-08-06 CN disclosed
CN-113226990-A Method for producing nanoparticles comprising iron oxide-containing metal particles to which one or more hydrophilic ligands are coordinately bound 安斯泰来制药株式会社 2021-08-06 CN disclosed
US-11008345-B2 Boron-containing small molecules ANACOR PHARMACEUTICALS, INC. (US) 2021-05-18 US disclosed
US-11008345-B2 Boron-containing small molecules ANACOR PHARMACEUTICALS, INC. (US) 2021-05-18 US disclosed
CN-108610356-B Benzoxaborole derivatives for the treatment of bacterial infections 阿纳科制药公司 2021-02-26 CN disclosed
WO-2020138404-A1 METHOD FOR PRODUCING NANOPARTICLES INCLUDING METAL PARTICLES CONTAINING IRON OXIDE HAVING AT LEAST ONE HYDROPHILIC LIGAND COORDINATED THERETO アステラス製薬株式会社 2020-07-02 WO disclosed
CN-103140228-A Benzoxaborole derivatives for the treatment of bacterial infections ANACOR PHARMACEUTICALS INC 2013-06-05 CN disclosed
US-20120115813-A1 BORON-CONTAINING SMALL MOLECULES ANACOR PHARMACEUTICALS, INC. (US) 2012-05-10 US disclosed
US-20120115813-A1 BORON-CONTAINING SMALL MOLECULES ANACOR PHARMACEUTICALS, INC. (US) 2012-05-10 US disclosed
US-20120115813-A1 BORON-CONTAINING SMALL MOLECULES ANACOR PHARMACEUTICALS, INC. (US) 2012-05-10 US disclosed
WO-2012033858-A2 BORON-CONTAINING SMALL MOLECULES ANACOR PHARMACEUTICALS, INC. (US) 2012-03-15 WO disclosed
WO-2012033858-A2 BORON-CONTAINING SMALL MOLECULES ANACOR PHARMACEUTICALS, INC. (US) 2012-03-15 WO disclosed
US-7091220-B2 Substituted indole Mannich bases GRUENENTHAL GMBH (DE) 2006-08-15 US disclosed
CN-1219763-C Substituted indole mannich bases GRUENENTHAL GMBH (DE) 2005-09-21 CN disclosed
CN-1413192-A Substituted indole mannich bases GRUENENTHAL GMBH (DE) 2003-04-23 CN disclosed
US-20030060497-A1 Subtituted indole mannich bases GRUENENTHAL GMBH (DE) 2003-03-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030060497-A1 Subtituted indole mannich bases TPH1, IDO1, TPH2 CA1 2887/4885CA2 2406/4885ALDH1A1 667/4885
US-20220089455-A1 METHOD FOR PRODUCING NANOPARTICLE HAVING METAL PARTICLE WHICH CONTAINS IRON OXIDE TO WHICH ONE OR MORE HYDROPHILIC LIGANDS ARE COORDINATION BONDED FTH1, HAMP, TFRC CA1 934/4885CA2 1788/4885ALDH1A1 2870/4885
US-11008345-B2 Boron-containing small molecules BCL6B, BTD, BROX CA1 4452/4885CA2 1021/4885ALDH1A1 4256/4885
US-20120115813-A1 BORON-CONTAINING SMALL MOLECULES BCL6B, BTD, BROX CA1 4452/4885CA2 1021/4885ALDH1A1 4256/4885
US-20220184236-A1 NANOPARTICLE, CONTRAST AGENT FOR MAGNETIC RESONANCE IMAGING COMPRISING SAME AND ZWITTERIONIC LIGAND COMPOUND CD47, LPAR3, NMRAL1 CA1 555/4885CA2 372/4885ALDH1A1 3785/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.