SCHEMBL4537343

SCHEMBL4537343

O=C(CC1CCCN(S(=O)(=O)c2ccc(Cl)cc2)C1)NC12CC3CC(CC(C3)C1)C2

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.59
HTT P42858 2/20 0.59
NPSR1 Q6W5P4 2/20 0.59
TSHR P16473 1/20 0.59
ALOX12 P18054 1/20 0.59
EPHX2 P34913 1/20 0.49
EPHX1 P07099 3/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
USP2 O75604 1/20 0.46
ALDH1A1 P00352 2/20 0.46
POLB P06746 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
DPP4 P27487 1/20 0.45
GAA P10253 1/20 0.45
HPGD P15428 2/20 0.44
KDM4E B2RXH2 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
FKBP1A P62942 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4536776 0.95 LMNA (0.62) LMNAHTTNPSR1TSHRALOX12
SCHEMBL4530361 0.90 CYP3A4 (0.59) LMNAHTTNPSR1TSHRALOX12
SCHEMBL4537575 0.90 ALDH1A1 (0.49) LMNAHTTNPSR1TSHRALOX12
SCHEMBL4537427 0.90 SMN1; SMN2 (0.52) LMNAHTTNPSR1TSHRALOX12
SCHEMBL4536605 0.89 LMNA (0.67) LMNAHTTNPSR1TSHRALOX12
SCHEMBL4539317 0.89 HSD11B1 (0.49) LMNAHTTNPSR1TSHRALOX12
SCHEMBL4539395 0.88 LMNA (0.47) LMNAHTTNPSR1TSHRALOX12
SCHEMBL4537319 0.87 ALDH1A1 (0.52) LMNAHTTNPSR1TSHREPHX1
SCHEMBL4537389 0.87 HTT (0.46) LMNAHTTNPSR1TSHRALOX12
SCHEMBL8060768 0.86 LMNA (0.57) LMNAHTTNPSR1TSHRALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed