SCHEMBL4536776

SCHEMBL4536776

O=C(CC1CCN(S(=O)(=O)c2ccc(Cl)cc2)C1)NC12CC3CC(CC(C3)C1)C2

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.62
HTT P42858 2/20 0.62
NPSR1 Q6W5P4 2/20 0.62
TSHR P16473 1/20 0.62
ALOX12 P18054 1/20 0.62
EPHX2 P34913 1/20 0.52
EPHX1 P07099 2/20 0.49
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 1/20 0.47
HPGD P15428 1/20 0.47
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.45
CYP3A4 P08684 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CNR1 P21554 1/20 0.42
USP2 O75604 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4537343 0.95 LMNA (0.59) LMNAHTTNPSR1TSHRALOX12
SCHEMBL4536605 0.94 LMNA (0.67) LMNAHTTNPSR1TSHRALOX12
SCHEMBL4539274 0.89 CYP3A4 (0.51) LMNAHTTNPSR1TSHRALOX12
SCHEMBL4535944 0.89 EPHX1 (0.52) LMNAHTTNPSR1TSHRALOX12
SCHEMBL4540431 0.89 NPC1 (0.55) LMNAHTTNPSR1TSHRALOX12
SCHEMBL4539809 0.88 HSD11B1 (0.52) LMNAHTTNPSR1TSHRALOX12
SCHEMBL8053303 0.88 HSD11B1 (0.52) LMNAHTTNPSR1TSHRALOX12
SCHEMBL4543052 0.88 NPC1 (0.48) LMNAHTTNPSR1TSHRALOX12
SCHEMBL4542516 0.88 LMNA (0.49) LMNAHTTNPSR1TSHRALOX12
SCHEMBL4540032 0.87 PKM (0.51) LMNAHTTNPSR1TSHRALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed