SCHEMBL4539756

SCHEMBL4539756

O=C(NCC1CCN(S(=O)(=O)c2ccccc2Cl)C1)[C]1CCCCCCC1.[CH2].[CH2]

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC10 Q969S8 1/20 0.50
HDAC11 Q96DB2 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
HDAC9 Q9UKV0 1/20 0.50
HDAC5 Q9UQL6 1/20 0.50
FAAH O00519 5/20 0.48
EPHX2 P34913 3/20 0.47
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 3/20 0.42
HSD11B1 P28845 1/20 0.42
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
ACLY P53396 1/20 0.41
MMP2 P08253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4538131 0.96 HDAC3 (0.46) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4542825 0.95 HDAC3 (0.53) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4537991 0.93 HDAC3 (0.45) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4541327 0.90 HDAC3 (0.51) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4537385 0.88 KMT2A (0.43) EPHX2KMT2AALDH1A1ACLY
SCHEMBL4533116 0.88 EPHX2 (0.50) EPHX2KMT2AALDH1A1
SCHEMBL4531620 0.86 HSD11B1 (0.58) EPHX2KMT2AALDH1A1HSD11B1
SCHEMBL4537189 0.86 FAAH (0.49) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4539751 0.85 ATM (0.50) ALDH1A1HSD11B1HTR2AHTR2C
SCHEMBL4542832 0.85 ALDH1A1 (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed